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BAY-6035

Product Name
BAY-6035
CAS No.
2247890-13-5
Chemical Name
BAY-6035
Synonyms
BAY-6035;BAY-6035, 10 mM in DMSO;inhibit,BAY-6035,Histone Methyltransferase,MEKK2,BAY6035,Inhibitor,BAY 6035,SMYD3,methylation;(2S)-1-(3-azabicyclo[3.1.0]hexane-3-carbonyl)-N-(2-cyclopropylethyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzodiazepine-7-carboxamide;(2S)-1-(3-Azabicyclo[3.1.0]hex-3-ylcarbonyl)-N-(2-cyclopropylethyl)-2,3,4,5-tetrahydro-2-methyl-4-oxo-1H-1,5-benzodiazepine-7-carboxamide;(2S)-1-{3-azabicyclo[3.1.0]hexane-3-carbonyl}-N-(2-cyclopropylethyl)-2-methyl-4-oxo-2,3,4,5-tetrahydro-1H-1,5-benzodiazepine-7-carboxamide;1H-1,5-Benzodiazepine-7-carboxamide, 1-(3-azabicyclo[3.1.0]hex-3-ylcarbonyl)-N-(2-cyclopropylethyl)-2,3,4,5-tetrahydro-2-methyl-4-oxo-, (2S)-;(2S)-1-(3-Azabicyclo[3.1.0]hexane-3-carbonyl)-N-(2-cyclopropylethyl)-2-methyl-4-oxo-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepine-7-carboxamide
CBNumber
CB35867500
Molecular Formula
C22H28N4O3
Formula Weight
396.48
MOL File
2247890-13-5.mol
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BAY-6035 Property

storage temp. 
Store at -20°C
solubility 
DMSO:39.65(Max Conc. mg/mL);100.0(Max Conc. mM)
Ethanol:39.65(Max Conc. mg/mL);100.0(Max Conc. mM)
form 
A crystalline solid
color 
White to off-white
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Hazard and Precautionary Statements (GHS)

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N-Bromosuccinimide Price

Cayman Chemical
Product number
25925
Product name
BAY-6035
Packaging
1mg
Price
$32
Updated
2024/03/01
Cayman Chemical
Product number
25925
Product name
BAY-6035
Packaging
5mg
Price
$109
Updated
2024/03/01
Cayman Chemical
Product number
25925
Product name
BAY-6035
Packaging
10mg
Price
$199
Updated
2024/03/01
Tocris
Product number
6561
Product name
BAY6035
Purity
≥98%(HPLC)
Packaging
25
Price
$360
Updated
2021/12/16
AK Scientific
Product number
0867EN
Product name
(2S)-1-(3-Azabicyclo[3.1.0]hexane-3-carbonyl)-N-(2-cyclopropylethyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzodiazepine-7-carboxamide
Packaging
1mg
Price
$133
Updated
2021/12/16
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BAY-6035 Chemical Properties,Usage,Production

Description

BAY 6035 is a potent and selective SMYD3 inhibitor.

in vitro

BAY-6035 specifically inhibited the methylation of MAP3K2 by SMYD3 in a cellular mechanistic assay with an IC50 <100 nM._x000D_ _x000D_ Reference: SLAS Discov. 2021 Jun 21:24725552211019409. https://journals.sagepub.com/doi/10.1177/24725552211019409?url_ver=Z39.88-2003&rfr_id=ori:rid:crossref.org&rfr_dat=cr_pub%20%200pubmed

target

BAY-6035 is a SMYD3 inhibitor.

storage

Store at -20°C

BAY-6035 Preparation Products And Raw materials

Raw materials

Preparation Products

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BAY-6035 Suppliers

China 27 United States 4 Global 31
TargetMol Chemicals Inc.
Tel
+1-781-999-5354 +1-00000000000
Email
marketing@targetmol.com
Country
United States
ProdList
32161
Advantage
58
Aladdin Scientific
Tel
+1-+1(833)-552-7181
Email
sales@aladdinsci.com
Country
United States
ProdList
52924
Advantage
58
TargetMol Chemicals Inc.
Tel
Email
support@targetmol.com
Country
United States
ProdList
38631
Advantage
58
Cayman Chemical Company
Tel
--
Fax
--
Email
cayman@caymanchem.com
Country
United States
ProdList
6213
Advantage
81

2247890-13-5, BAY-6035Related Search:


  • BAY-6035
  • 1H-1,5-Benzodiazepine-7-carboxamide, 1-(3-azabicyclo[3.1.0]hex-3-ylcarbonyl)-N-(2-cyclopropylethyl)-2,3,4,5-tetrahydro-2-methyl-4-oxo-, (2S)-
  • inhibit,BAY-6035,Histone Methyltransferase,MEKK2,BAY6035,Inhibitor,BAY 6035,SMYD3,methylation
  • (2S)-1-(3-azabicyclo[3.1.0]hexane-3-carbonyl)-N-(2-cyclopropylethyl)-2-methyl-4-oxo-3,5-dihydro-2H-1,5-benzodiazepine-7-carboxamide
  • (2S)-1-(3-Azabicyclo[3.1.0]hex-3-ylcarbonyl)-N-(2-cyclopropylethyl)-2,3,4,5-tetrahydro-2-methyl-4-oxo-1H-1,5-benzodiazepine-7-carboxamide
  • (2S)-1-(3-Azabicyclo[3.1.0]hexane-3-carbonyl)-N-(2-cyclopropylethyl)-2-methyl-4-oxo-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepine-7-carboxamide
  • (2S)-1-{3-azabicyclo[3.1.0]hexane-3-carbonyl}-N-(2-cyclopropylethyl)-2-methyl-4-oxo-2,3,4,5-tetrahydro-1H-1,5-benzodiazepine-7-carboxamide
  • BAY-6035, 10 mM in DMSO
  • 2247890-13-5