ChemicalBook > CAS DataBase List > (2S)-2-AMINOPROPYL ESTER N2-[[2-(2-NAPHTHALENYL)-1H-BENZ[G]INDOL-3-YL]ACETYL]-D-LYSINE

(2S)-2-AMINOPROPYL ESTER N2-[[2-(2-NAPHTHALENYL)-1H-BENZ[G]INDOL-3-YL]ACETYL]-D-LYSINE

Product Name
(2S)-2-AMINOPROPYL ESTER N2-[[2-(2-NAPHTHALENYL)-1H-BENZ[G]INDOL-3-YL]ACETYL]-D-LYSINE
CAS No.
217480-27-8
Chemical Name
(2S)-2-AMINOPROPYL ESTER N2-[[2-(2-NAPHTHALENYL)-1H-BENZ[G]INDOL-3-YL]ACETYL]-D-LYSINE
Synonyms
818;L-817;L-817,818;L 817,818,L817,818;N2-[[2-(2-Naphthalenyl)-1H-benz[g]indol-3-yl]acetyl-D-lysine(2S)-2-aminopropylester;(2S)-2-AMINOPROPYL ESTER N2-[[2-(2-NAPHTHALENYL)-1H-BENZ[G]INDOL-3-YL]ACETYL]-D-LYSINE;D-Lysine, N2-[2-[2-(2-naphthalenyl)-1H-benz[g]indol-3-yl]acetyl]-, (2S)-2-aminopropyl ester
CBNumber
CB42453419
Molecular Formula
C33H36N4O3
Formula Weight
536.66
MOL File
217480-27-8.mol
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(2S)-2-AMINOPROPYL ESTER N2-[[2-(2-NAPHTHALENYL)-1H-BENZ[G]INDOL-3-YL]ACETYL]-D-LYSINE Property

Boiling point:
827.9±65.0 °C(Predicted)
Density 
1.235±0.06 g/cm3(Predicted)
storage temp. 
Store at -20°C
solubility 
Soluble to 100 mM in DMSO
form 
Powder
pka
14.07±0.46(Predicted)
color 
White to off-white
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Hazard and Precautionary Statements (GHS)

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N-Bromosuccinimide Price

Tocris
Product number
1980
Product name
L-817,818
Purity
≥99%(HPLC)
Packaging
10
Price
$318
Updated
2021/12/16
Usbiological
Product number
255644
Product name
L-817,818
Packaging
10mg
Price
$588
Updated
2021/12/16
ApexBio Technology
Product number
B6905
Product name
L-817,818
Packaging
10mg
Price
$480
Updated
2021/12/16
American Custom Chemicals Corporation
Product number
API0009981
Product name
L-817,818
Purity
95.00%
Packaging
5MG
Price
$497.19
Updated
2021/12/16
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(2S)-2-AMINOPROPYL ESTER N2-[[2-(2-NAPHTHALENYL)-1H-BENZ[G]INDOL-3-YL]ACETYL]-D-LYSINE Chemical Properties,Usage,Production

Uses

L-817,818 is a potent sst5 agonist.

Biological Activity

Potent and selective somatostatin sst 5 receptor agonist. K i values are 0.4, 3.3, 52, 64 and 82 nM for cloned human sst 5 , sst 1 , sst 2 , sst 3 and sst 4 receptors respectively. Inhibits growth hormone release from rat pituitary cells (EC 50 = 3.1 nM) and insulin release from mouse pancreatic islets (EC 50 = 0.3 nM) in vitro .

storage

Store at -20°C

(2S)-2-AMINOPROPYL ESTER N2-[[2-(2-NAPHTHALENYL)-1H-BENZ[G]INDOL-3-YL]ACETYL]-D-LYSINE Preparation Products And Raw materials

Raw materials

Preparation Products

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(2S)-2-AMINOPROPYL ESTER N2-[[2-(2-NAPHTHALENYL)-1H-BENZ[G]INDOL-3-YL]ACETYL]-D-LYSINE Suppliers

CHINA 12 United Kingdom 1 United States 5 USA 1 Global 19
Tocris Bioscience
Tel
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Fax
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Email
customerservice@tocris.co.uk
Country
United Kingdom
ProdList
5726
Advantage
77

217480-27-8, (2S)-2-AMINOPROPYL ESTER N2-[[2-(2-NAPHTHALENYL)-1H-BENZ[G]INDOL-3-YL]ACETYL]-D-LYSINERelated Search:

2-(2-NAPHTHYL)INDOLE INDOLE-3-ACETYL GLYCINE AC-D-LYS-OH (2S)-2-AMINOPROPYL ESTER N2-[[2-(2-NAPHTHALENYL)-1H-BENZ[G]INDOL-3-YL]ACETYL]-D-LYSINE

  • (2S)-2-AMINOPROPYL ESTER N2-[[2-(2-NAPHTHALENYL)-1H-BENZ[G]INDOL-3-YL]ACETYL]-D-LYSINE
  • L-817,818
  • N2-[[2-(2-Naphthalenyl)-1H-benz[g]indol-3-yl]acetyl-D-lysine(2S)-2-aminopropylester
  • D-Lysine, N2-[2-[2-(2-naphthalenyl)-1H-benz[g]indol-3-yl]acetyl]-, (2S)-2-aminopropyl ester
  • 818
  • L-817
  • L 817,818,L817,818
  • 217480-27-8