ChemicalBook > CAS DataBase List > (8R)-8-ETHYL-1,4,7,8-TETRAHYDRO-4-5H-IMIDAZO[2,1-I]PURIN-5-ONE
(8R)-8-ETHYL-1,4,7,8-TETRAHYDRO-4-5H-IMIDAZO[2,1-I]PURIN-5-ONE
- Product Name
- (8R)-8-ETHYL-1,4,7,8-TETRAHYDRO-4-5H-IMIDAZO[2,1-I]PURIN-5-ONE
- CAS No.
- 444717-56-0
- Chemical Name
- (8R)-8-ETHYL-1,4,7,8-TETRAHYDRO-4-5H-IMIDAZO[2,1-I]PURIN-5-ONE
- Synonyms
- PSB 11 HYDROCHLORIDE;(8R)-8-ETHYL-1,4,7,8-TETRAHYDRO-4-5H-IMIDAZO[2,1-I]PURIN-5-ONE;(8R)-8-ETHYL-1,4,7,8-TETRAHYDRO-4-5H-IMIDAZO[2,1-I]PURIN-5-ONE HYDROCHLORIDE;5H-Imidazo[2,1-i]purin-5-one, 8-ethyl-3,4,7,8-tetrahydro-4-methyl-2-phenyl-, (8R)-
- CBNumber
- CB4332396
- Molecular Formula
- C16H17N5O
- Formula Weight
- 295.34
- MOL File
- 444717-56-0.mol
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(8R)-8-ETHYL-1,4,7,8-TETRAHYDRO-4-5H-IMIDAZO[2,1-I]PURIN-5-ONE Property
- storage temp.
- Store at +4°C
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N-Bromosuccinimide Price
Tocris
- Product number
- 2012
- Product name
- PSB11hydrochloride
- Purity
- ≥98%(HPLC)
- Packaging
- 10
- Price
- $189
- Updated
- 2021/12/16
Tocris
- Product number
- 2012
- Product name
- PSB11hydrochloride
- Purity
- ≥98%(HPLC)
- Packaging
- 50
- Price
- $744
- Updated
- 2021/12/16
Usbiological
- Product number
- 256351
- Product name
- PSB 11 hydrochloride
- Packaging
- 10mg
- Price
- $466
- Updated
- 2021/12/16
American Custom Chemicals Corporation
- Product number
- API0009889
- Product name
- PSB 11 HYDROCHLORIDE
- Purity
- 95.00%
- Packaging
- 5MG
- Price
- $503.22
- Updated
- 2021/12/16
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(8R)-8-ETHYL-1,4,7,8-TETRAHYDRO-4-5H-IMIDAZO[2,1-I]PURIN-5-ONE Chemical Properties,Usage,Production
Uses
PSB 11 Hydrochloride is a potent and selective antagonist of Adenosine receptor A3-R.
Biological Activity
Potent and selective antagonist for the human adenosine A 3 receptor, with low affinity for the rat A 3 receptor (K i values are 2.3 and > 10000 nM respectively). Displays > 1000-fold selectivity over human A 1 and A 2A receptors (K i values are 4.1 and 3.3 μ M respectively) and > 180-fold selectivity over rat A 1 , rat A 2A and mouse A 2B receptors. Acts as an inverse agonist in the [ 35 S]GTP γ S binding assay in hA 3 -CHO cells (IC 50 = 36 nM).
(8R)-8-ETHYL-1,4,7,8-TETRAHYDRO-4-5H-IMIDAZO[2,1-I]PURIN-5-ONE Preparation Products And Raw materials
Raw materials
Preparation Products
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(8R)-8-ETHYL-1,4,7,8-TETRAHYDRO-4-5H-IMIDAZO[2,1-I]PURIN-5-ONE Suppliers
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- 821-50328103-801 18930552037
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