GSK4028

Product Name: GSK4028
CAS No.: 2079886-19-2
Chemical Name: GSK4028
Synonyms: GSK4028;3(2H)-Pyridazinone, 4-bromo-2-methyl-5-[[(3S,5S)-1-methyl-5-phenyl-3-piperidinyl]amino]-
CBNumber: CB44797067
Molecular Formula: C17H21BrN4O
Formula Weight: 377.28
MOL File: 2079886-19-2.mol

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GSK4028 Property

Boiling point:: 450.3±55.0 °C(Predicted)
Density: 1.45±0.1 g/cm3(Predicted)
storage temp.: Store at -20°C
solubility: Soluble in DMSO
form: Solid
pka: 9.58±0.10(Predicted)
color: Light yellow to yellow

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Hazard and Precautionary Statements (GHS)

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N-Bromosuccinimide Price

ChemScene

Product number: CS-0058953
Product name: GSK4028
Purity: 98.11%
Packaging: 5mg
Price: $550
Updated: 2021/12/16

ChemScene

Product number: CS-0058953
Product name: GSK4028
Purity: 98.11%
Packaging: 10mg
Price: $850
Updated: 2021/12/16

ChemScene

Product number: CS-0058953
Product name: GSK4028
Purity: 98.11%
Packaging: 25mg
Price: $1750
Updated: 2021/12/16

ChemScene

Product number: CS-0058953
Product name: GSK4028
Purity: 98.11%
Packaging: 50mg
Price: $2750
Updated: 2021/12/16

ChemScene

Product number: CS-0058953
Product name: GSK4028
Purity: 98.11%
Packaging: 100mg
Price: $3950
Updated: 2021/12/16

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GSK4028 Chemical Properties,Usage,Production

Description

GSK4028 is the enantiomeric negative control of GSK4027, which is a PCAF/GCN5 bromodomain chemical probe, the pIC50 of GSK4028 is 4.9 in a time-resolved fluorescence resonance energy transfer (TR-FRET) assay.

GSK4028 is the enantiomeric negative control of GSK4027, which is a PCAF/GCN5 bromodomain chemical probe, the pIC50 of GSK4028 is 4.9. GSK4028 also demonstrates potency toward BRD4 BD1 and BRD9 inTR-FRET assay with pIC50s of <4.3 and 4.5±0.13, respectively[1].

References

[1]. Humphreys PG, et al. Discovery of a Potent, Cell Penetrant, and Selective p300/CBP-Associated Factor (PCAF)/General Control Nonderepressible 5 (GCN5) Bromodomain Chemical Probe. J Med Chem. 2017 Jan 26;60(2):695-709.

GSK4028 Preparation Products And Raw materials

Raw materials

Preparation Products

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GSK4028 Suppliers

China 10 United States 5 Global 15

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2079886-19-2, GSK4028Related Search:

GSK4028

3(2H)-Pyridazinone, 4-bromo-2-methyl-5-[[(3S,5S)-1-methyl-5-phenyl-3-piperidinyl]amino]-

2079886-19-2