ChemicalBook > CAS DataBase List > 8-ETHYL-1,4,7,8-TETRAHYDRO-4-METHYL-2-(2,3,5-TRICHLOROPHENYL)-5H-IMIDAZO[2,1-I]PURIN-5-ONE MONOHYDROCHLORIDE
8-ETHYL-1,4,7,8-TETRAHYDRO-4-METHYL-2-(2,3,5-TRICHLOROPHENYL)-5H-IMIDAZO[2,1-I]PURIN-5-ONE MONOHYDROCHLORIDE
- Product Name
- 8-ETHYL-1,4,7,8-TETRAHYDRO-4-METHYL-2-(2,3,5-TRICHLOROPHENYL)-5H-IMIDAZO[2,1-I]PURIN-5-ONE MONOHYDROCHLORIDE
- CAS No.
- 591771-91-4
- Chemical Name
- 8-ETHYL-1,4,7,8-TETRAHYDRO-4-METHYL-2-(2,3,5-TRICHLOROPHENYL)-5H-IMIDAZO[2,1-I]PURIN-5-ONE MONOHYDROCHLORIDE
- Synonyms
- PSB 10;PSB 10 HYDROCHLORIDE;8-ETHYL-1,4,7,8-TETRAHYDRO-4-METHYL-2-(2,3,5-TRICHLOROPHENYL)-5H-IMIDAZO[2,1-I]PURIN-5-ONE MONOHYDROCHLORIDE
- CBNumber
- CB4842011
- Molecular Formula
- C16H14Cl3N5O.ClH
- Formula Weight
- 435.141
- MOL File
- 591771-91-4.mol
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8-ETHYL-1,4,7,8-TETRAHYDRO-4-METHYL-2-(2,3,5-TRICHLOROPHENYL)-5H-IMIDAZO[2,1-I]PURIN-5-ONE MONOHYDROCHLORIDE Property
- storage temp.
- Desiccate at +4°C
- solubility
- Soluble to 25 mM in DMSO and to 10 mM in ethanol
- form
- Powder
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N-Bromosuccinimide Price
Tocris
- Product number
- 2010
- Product name
- PSB10hydrochloride
- Purity
- ≥98%(HPLC)
- Packaging
- 10
- Price
- $212
- Updated
- 2021/12/16
Tocris
- Product number
- 2010
- Product name
- PSB10hydrochloride
- Purity
- ≥98%(HPLC)
- Packaging
- 50
- Price
- $891
- Updated
- 2021/12/16
ApexBio Technology
- Product number
- B6923
- Product name
- PSB10hydrochloride
- Packaging
- 50mg
- Price
- $1322
- Updated
- 2021/12/16
ApexBio Technology
- Product number
- B6923
- Product name
- PSB10hydrochloride
- Packaging
- 10mg
- Price
- $314
- Updated
- 2021/12/16
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8-ETHYL-1,4,7,8-TETRAHYDRO-4-METHYL-2-(2,3,5-TRICHLOROPHENYL)-5H-IMIDAZO[2,1-I]PURIN-5-ONE MONOHYDROCHLORIDE Chemical Properties,Usage,Production
Biological Activity
Potent and highly selective antagonist for the human adenosine A 3 receptor, with low affinity for the rat A 3 receptor (K i values are 0.44 and > 17000 nM respectively). Displays > 3800-fold selectivity over human A 1 , A 2A and A 2B receptors (K i values are 4.1, 3.3 and 30 μ M respectively) and > 1800-fold selectivity over rat A 1 and A 2A receptors. Acts as an inverse agonist in the [ 35 S]GTP γ S binding assay in hA 3 -CHO cells (IC 50 = 4 nM). Produces thermal hyperalgesia in mice in vivo .
storage
Desiccate at +4°C
8-ETHYL-1,4,7,8-TETRAHYDRO-4-METHYL-2-(2,3,5-TRICHLOROPHENYL)-5H-IMIDAZO[2,1-I]PURIN-5-ONE MONOHYDROCHLORIDE Preparation Products And Raw materials
Raw materials
Preparation Products
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8-ETHYL-1,4,7,8-TETRAHYDRO-4-METHYL-2-(2,3,5-TRICHLOROPHENYL)-5H-IMIDAZO[2,1-I]PURIN-5-ONE MONOHYDROCHLORIDE Suppliers
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