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Fedovapagon

Product Name
Fedovapagon
CAS No.
347887-36-9
Chemical Name
Fedovapagon
Synonyms
Fedovapagon;Fedovapagon, 10 mM in DMSO;(S)-N2,N2-Dimethyl-N1-(2-methyl-4-(2,3,4,5-tetrahydro-1H-benzo[b]azepine-1-carbonyl)benzyl)pyrrolidine-1,2-dicarboxamide;1,2-Pyrrolidinedicarboxamide, N2,N2-dimethyl-N1-[[2-methyl-4-[(2,3,4,5-tetrahydro-1H-1-benzazepin-1-yl)carbonyl]phenyl]methyl]-, (2S)-
CBNumber
CB52627882
Molecular Formula
C27H34N4O3
Formula Weight
462.58
MOL File
347887-36-9.mol
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Fedovapagon Property

Boiling point:
740.0±60.0 °C(Predicted)
Density 
1.203±0.06 g/cm3(Predicted)
storage temp. 
Store at -20°C
solubility 
DMSO: ≥ 125 mg/mL (270.22 mM)
form 
Solid
pka
13.38±0.40(Predicted)
color 
Off-white to light yellow
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Warning
Hazard statements

H302Harmful if swallowed

H315Causes skin irritation

H319Causes serious eye irritation

H335May cause respiratory irritation

Precautionary statements

P261Avoid breathing dust/fume/gas/mist/vapours/spray.

P280Wear protective gloves/protective clothing/eye protection/face protection.

P301+P312IF SWALLOWED: call a POISON CENTER or doctor/physician IF you feel unwell.

P302+P352IF ON SKIN: wash with plenty of soap and water.

P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

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N-Bromosuccinimide Price

TRC
Product number
F229080
Product name
Fedovapagon
Packaging
1g
Price
$1320
Updated
2021/12/16
ChemScene
Product number
CS-0003613
Product name
Fedovapagon
Purity
99.03%
Packaging
5mg
Price
$140
Updated
2021/12/16
ChemScene
Product number
CS-0003613
Product name
Fedovapagon
Purity
99.03%
Packaging
10mg
Price
$220
Updated
2021/12/16
American Custom Chemicals Corporation
Product number
API0013908
Product name
FEDOVAPAGON
Purity
95.00%
Packaging
5MG
Price
$320.1
Updated
2021/12/16
ChemScene
Product number
CS-0003613
Product name
Fedovapagon
Purity
99.03%
Packaging
50mg
Price
$850
Updated
2021/12/16
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Fedovapagon Chemical Properties,Usage,Production

Uses

Fedovapagon is a potent, nonpeptidic vasopressin V2 receptor agonists.

in vivo

Fedovapagon (1 mg/kg, oral administration) inhibits urine output with 81% inhibition rate in rats[1].

Animal Model:Brattleboro rats[1]
Dosage:1 mg/kg, 3 mg/kg
Administration:Oral administration
Result:Reduced urine volume with almost full inhibition of urine output for 2 h.
Returned the urine to normal levels 5 h after dosing.

IC 50

V2 Receptor; V2 Receptor: 24 nM (EC50)

Fedovapagon Preparation Products And Raw materials

Raw materials

Preparation Products

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Fedovapagon Suppliers

China 27 India 1 United States 3 USA 1 Global 32
ShangHai Wisacheam Pharmaceutical Co., Ltd.
Tel
13817485796
Fax
QQ:895624079
Email
tim@wisacheampharm.com
Country
China
ProdList
3592
Advantage
58
Shanghai EFE Biological Technology Co., Ltd.
Tel
021-65675885 18964387627
Fax
021-65675885
Email
info@efebio.com
Country
China
ProdList
9803
Advantage
58
Shanghai Biopharmaleader Co., Ltd.
Tel
+86 18721201413
Fax
+86 (21) 5775-8967
Email
sales@biopharmaleader.com
Country
China
ProdList
1720
Advantage
58
TargetMol Chemicals Inc.
Tel
+1-781-999-5354; +17819995354
Email
marketing@targetmol.com
Country
United States
ProdList
32435
Advantage
58
ChemeGen(Shanghai) Biotechnology Co.,Ltd.
Tel
18818260767
Fax
QQ 3610331285
Email
sales@chemegen.com
Country
China
ProdList
11218
Advantage
58
Wuhan Dingxintong Pharmaceutical Co. , Ltd.
Tel
15871722230
Fax
2796190295
Email
15871722230@163.com
Country
China
ProdList
4686
Advantage
58
ShangHai ChuanQian Chemcial Technique Centre
Tel
15869524721
Email
3525679403@qq.com
Country
China
ProdList
4989
Advantage
58
Energy Chemical
Tel
021-58432009 400-005-6266
Fax
021-58436166
Email
marketing@energy-chemical.com
Country
China
ProdList
44918
Advantage
58
Bide Pharmatech Ltd.
Tel
400-1647117 13681763483
Email
product02@bidepharm.com
Country
China
ProdList
62220
Advantage
58
TargetMol Chemicals Inc.
Tel
4008200310
Email
marketing@tsbiochem.com
Country
China
ProdList
24961
Advantage
58

347887-36-9, FedovapagonRelated Search:


  • Fedovapagon
  • 1,2-Pyrrolidinedicarboxamide, N2,N2-dimethyl-N1-[[2-methyl-4-[(2,3,4,5-tetrahydro-1H-1-benzazepin-1-yl)carbonyl]phenyl]methyl]-, (2S)-
  • (S)-N2,N2-Dimethyl-N1-(2-methyl-4-(2,3,4,5-tetrahydro-1H-benzo[b]azepine-1-carbonyl)benzyl)pyrrolidine-1,2-dicarboxamide
  • Fedovapagon, 10 mM in DMSO
  • 347887-36-9