TAS-102

Product Name: TAS-102
CAS No.: 733030-01-8
Chemical Name: TAS-102
Synonyms: TAS-102;TAS 102 (2:1);TAS102; TAS 102;TAS-102 (LONSURF);TAS-102(TIPIRACIL, TRIFLURIDINE);TAS-102 (Trifluridine/Tipiracil HCl);Trifluridine-tipiracil hydrochloride mixt.;Tipiracil hydrochloride-trifluridine mixt.;rifluridine-tipiracil hydrochloride mixture;TRIFLURIDINE-TIPIRACIL HYDROCHLORIDE MIXTURE
CBNumber: CB52667622
Molecular Formula: C19H23Cl2F3N6O7
Formula Weight: 575.32
MOL File: 733030-01-8.mol

More

Less

TAS-102 Property

Melting point:: 170-172°C
storage temp.: Hygroscopic, Refrigerator, under inert atmosphere
solubility: DMSO (Slightly, Heated, Sonicated), Methanol (Slightly)
form: Solid
color: White to Off-White
Stability:: Hygroscopic

More

Less

Hazard and Precautionary Statements (GHS)

Symbol(GHS)

Signal word

Warning

Hazard statements

H341Suspected of causing genetic defects

H351Suspected of causing cancer

Precautionary statements

P201Obtain special instructions before use.

P308+P313IF exposed or concerned: Get medical advice/attention.

More

Less

N-Bromosuccinimide Price

Sigma-Aldrich

Product number: SML2707
Product name: TAS-102
Purity: ≥98% (HPLC)
Packaging: 10MG
Price: $128.25
Updated: 2025/07/31

Cayman Chemical

Product number: 23932
Product name: TAS 102
Packaging: 5mg
Price: $50
Updated: 2023/01/06

Cayman Chemical

Product number: 23932
Product name: TAS 102
Packaging: 10mg
Price: $94
Updated: 2023/01/06

Cayman Chemical

Product number: 23932
Product name: TAS 102
Packaging: 25mg
Price: $207
Updated: 2023/01/06

Cayman Chemical

Product number: 23932
Product name: TAS 102
Packaging: 50mg
Price: $366
Updated: 2023/01/06

More

Less

TAS-102 Chemical Properties,Usage,Production

Uses

TAS 102 (Tipiracil-trifluridine) is a thymidine phosphorylase inhibitor used in chemotherapy treatment of advanced/recurring colorectal cancer.

Biological Activity

Anti cancer, Anti angiogenic

in vivo

Trifluridine/tipiracil hydrochloride mixture (150 mg/kg/day; p.o.; twice a day for 14 days) prevents body weight loss and reduces the relative tumor volume in colorectal cancer and gastric cancer mice models^[2].

Animal Model:	Male nude mice bearing KM12C, KM12C/5-FU, DLD-1, DLD-1/5-FU, and SC-2 cells^[2]
Dosage:	150 mg/kg/day
Administration:	p.o.; twice a day for 14 days
Result:	Prevented body weight loss and reduced the relative tumor volume in colorectal cancer and gastric cancer mice models.

TAS-102 Preparation Products And Raw materials

Raw materials

Preparation Products

More

Less

TAS-102 Suppliers

China 77 United States 11 Global 88

Shanghai Boyle Chemical Co., Ltd.

Tel
Fax: 86-21-57758967
Email: sales@boylechem.com
Country: China
ProdList: 2922
Advantage: 55

Dalian Meilun Biotech Co., Ltd.

Tel: 0411-62910999 13889544652
Email: sales@meilune.com
Country: China
ProdList: 4747
Advantage: 58

MedChemexpress LLC

Tel: 021-58955995
Fax: 609-228-5909
Email: sales@medchemexpress.cn
Country: United States
ProdList: 4861
Advantage: 58

ShangHai Caerulum Pharma Discovery Co., Ltd.

Tel: 18149758185
Email: sales-cpd@caerulumpharma.com
Country: China
ProdList: 3506
Advantage: 58

AdooQ Bioscience CHINA

Tel: 025-58849295 18951903616;
Fax: 025-68650336
Email: info@adooq.cn
Country: China
ProdList: 2990
Advantage: 60

Shanghai Lollane Biological Technology Co.,Ltd.

Tel: 021-52996696，15000506266 15000506266
Fax: +86-21-52996696
Country: China
ProdList: 4757
Advantage: 55

SPIRO PHARMA

Tel
Fax: -
Email: eric_feng1954@126.com
Country: China
ProdList: 9248
Advantage: 55

Shanghai YuanYe Biotechnology Co., Ltd.

Tel: 021-61312847; 18021002903
Fax: QQ:3008007432
Email: 3008007409@qq.com
Country: China
ProdList: 71826
Advantage: 60

Shanghai SuperLan Chemcial Technique Centre

Tel: 0-2022843681 15618226720
Fax: +86-21-51601218
Email: chaolaichem@foxmail.com
Country: China
ProdList: 12476
Advantage: 58

Beijing Solarbio Science & Tecnology Co., Ltd.

Tel: 010-50973130 18101056239
Email: 3193328036@qq.com
Country: China
ProdList: 29760
Advantage: 68

733030-01-8, TAS-102Related Search:

Futibatinib TAS6417 TAS0728 TAS-301 TAS-116

TAS-102

Tipiracil hydrochloride-trifluridine mixt.

TRIFLURIDINE-TIPIRACIL HYDROCHLORIDE MIXTURE

TAS-102(Tipiracil hydrochloride-trifluridine mixt)

Trifluridine-tipiracil hydrochloride mixt.

TAS-102(TIPIRACIL, TRIFLURIDINE)

TAS-102 (LONSURF)

TAS102; TAS 102

TAS 102 (2:1)

TAS-102 (Trifluridine/Tipiracil HCl)

inhibit,Thymidylate Synthase,Nucleoside Antimetabolite/Analog,oral,Inhibitor,FTD,DNA,nucleoside,antitumor,TPI,Trifluridine/tipiracil hydrochloride mixture

rifluridine-tipiracil hydrochloride mixture

1-((2R,4S,5R)-4-Hydroxy-5-(hydroxymethyl)tetrahydrofuran-2-yl)-5-(trifluoromethyl)pyrimidine-2,4(1H,3H)-dione mixt. with 5-chloro-6-((2-iminopyrrolidin-1-yl)methyl)pyrimidine-2,4(1H,3H)-dione (1:1) hydrochloride

Trifluridine/tipiracil hydrochloride mixture, 10 mM in DMSO

733030-01-8

C10H11F3N2O5C9H11ClN4O2HCl