Balovaptan

Product Name: Balovaptan
CAS No.: 1228088-30-9
Chemical Name: Balovaptan
Synonyms: RG7314;Balovaptan;RO-5285119;Balovaptan(RG7314);Balovaptan, 10 mM in DMSO;RG 7314,Vasopressin Receptor,RG-7314,inhibit,Inhibitor,Balovaptan;trans-8-chloro-5-methyl-1-[4-(pyridin-2-yloxy)cyclohexyl]-5,6-dihydro-4H-2,3,5,10b-tetraazabenzo[e]azulene;4H-[1,2,4]Triazolo[4,3-a][1,4]benzodiazepine, 8-chloro-5,6-dihydro-5-methyl-1-[trans-4-(2-pyridinyloxy)cyclohexyl]-;8-Chloro-5-methyl-1-((1r,4r)-4-(pyridin-2-yloxy)cyclohexyl)-5,6-dihydro-4H-benzo[f][1,2,4]triazolo[4,3-a][1,4]diazepine
CBNumber: CB54189016
Molecular Formula: C22H24ClN5O
Formula Weight: 409.91
MOL File: 1228088-30-9.mol

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Balovaptan Property

Boiling point:: 597.0±60.0 °C(Predicted)
Density: 1.39±0.1 g/cm3(Predicted)
storage temp.: Store at -20°C
solubility: DMSO: 62.5 mg/mL (152.47 mM)
form: Solid
pka: 5.52±0.20(Predicted)
color: White to off-white

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Hazard and Precautionary Statements (GHS)

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N-Bromosuccinimide Price

ChemScene

Product number: CS-0030526
Product name: Balovaptan
Purity: 99.18%
Packaging: 5mg
Price: $320
Updated: 2021/12/16

ChemScene

Product number: CS-0030526
Product name: Balovaptan
Purity: 99.18%
Packaging: 10mg
Price: $550
Updated: 2021/12/16

ChemScene

Product number: CS-0030526
Product name: Balovaptan
Purity: 99.18%
Packaging: 25mg
Price: $990
Updated: 2021/12/16

ChemScene

Product number: CS-0030526
Product name: Balovaptan
Purity: 99.18%
Packaging: 50mg
Price: $1650
Updated: 2021/12/16

ChemScene

Product number: CS-0030526
Product name: Balovaptan
Purity: 99.18%
Packaging: 100mg
Price: $2250
Updated: 2021/12/16

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Balovaptan Chemical Properties,Usage,Production

Uses

Balovaptan (RG7314) is an orally available, selective brain-penetrant vasopressin 1a (hV1a) receptor antagonist, with Kis of 1 and 39 nM for human (hV1a) and mouse (mV1a) receptors, and is used for the research of autism.

References

[1] Ratni H, et al. Discovery of highly selective brain-penetrant vasopressin 1a antagonists for the potential treatment of autism via a chemogenomic and scaffold hopping approach. J Med Chem. 2015 Mar 12;58(5):2275-89. DOI:10.1021/jm501745f

Balovaptan Preparation Products And Raw materials

Raw materials

Preparation Products

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Balovaptan Suppliers

China 39 United States 2 Global 41

Bide Pharmatech Ltd.

Tel: 400-400-164-7117 18317119277
Fax: +86-21-61629029
Email: product02@bidepharm.com
Country: China
ProdList: 40000
Advantage: 60

Shanghai Lollane Biological Technology Co.,Ltd.

Tel: 021-52996696，15000506266 15000506266
Fax: +86-21-52996696
Country: China
ProdList: 4800
Advantage: 55

NanJing Xienuo bio Co.,Ltd.

Tel: 025-84112752 13805181430
Fax: +86-25-84846489
Email: 154301870@qq.com
Country: China
ProdList: 998
Advantage: 55

Beijing Solarbio Science & Tecnology Co., Ltd.

Tel: 010-50973130 18101056239
Email: 3193328036@qq.com
Country: China
ProdList: 29662
Advantage: 68

Fan De(Beijing) Biotechnology Co., Ltd.

Tel: 15911056312
Email: liming@bio-fount.com
Country: China
ProdList: 9729
Advantage: 58

Nanjing Meihao Pharmaceutical Technology Co., Ltd.

Tel: meitaochem@126.com
Email: meitaochem@126.com
Country: China
ProdList: 19103
Advantage: 58

TargetMol Chemicals Inc.

Tel: +1-781-999-5354; +17819995354
Email: marketing@targetmol.com
Country: United States
ProdList: 32470
Advantage: 58

ChemeGen(Shanghai) Biotechnology Co.,Ltd.

Tel: 18818260767
Fax: QQ 3610331285
Email: sales@chemegen.com
Country: China
ProdList: 11218
Advantage: 58

Shanghai hongqu biomedical technology co. LTD

Tel: 88888888888
Email: hongquchem@qq.com
Country: China
ProdList: 5132
Advantage: 58

Wuhan Topule

Tel: +86-02787215551 +86-19945035818
Fax: 027-87215551
Email: 2936752263@qq.com
Country: China
ProdList: 7998
Advantage: 58

1228088-30-9, BalovaptanRelated Search:

Balovaptan

trans-8-chloro-5-methyl-1-[4-(pyridin-2-yloxy)cyclohexyl]-5,6-dihydro-4H-2,3,5,10b-tetraazabenzo[e]azulene

RG7314

4H-[1,2,4]Triazolo[4,3-a][1,4]benzodiazepine, 8-chloro-5,6-dihydro-5-methyl-1-[trans-4-(2-pyridinyloxy)cyclohexyl]-

Balovaptan(RG7314)

RG 7314,Vasopressin Receptor,RG-7314,inhibit,Inhibitor,Balovaptan

8-Chloro-5-methyl-1-((1r,4r)-4-(pyridin-2-yloxy)cyclohexyl)-5,6-dihydro-4H-benzo[f][1,2,4]triazolo[4,3-a][1,4]diazepine

Balovaptan, 10 mM in DMSO

RO-5285119

1228088-30-9