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morinamide

Product Name
morinamide
CAS No.
952-54-5
Chemical Name
morinamide
Synonyms
B 2310;morinamide;Morfazinamide;morphazinamide;N-(Morpholinomethyl)-2-pyrazinecarboxamide;2-Pyrazinecarboxamide, N-(4-morpholinylmethyl)-;pyrazine-2-carboxylic acid morpholin-4-ylmethyl-amide
CBNumber
CB5936067
Molecular Formula
C10H14N4O2
Formula Weight
222.24
MOL File
952-54-5.mol
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morinamide Property

Melting point:
118.5-119.5°
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Hazard and Precautionary Statements (GHS)

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N-Bromosuccinimide Price

TRC
Product number
M651765
Product name
Morphazinamide
Packaging
500mg
Price
$880
Updated
2021/12/16
American Custom Chemicals Corporation
Product number
API0011982
Product name
MORINAMIDE
Purity
95.00%
Packaging
50MG
Price
$2194.5
Updated
2021/12/16
American Custom Chemicals Corporation
Product number
API0011982
Product name
MORINAMIDE
Purity
95.00%
Packaging
5MG
Price
$816.75
Updated
2021/12/16
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morinamide Chemical Properties,Usage,Production

Originator

Morinamide,Bracco Industria Chimica S.p.A.

Uses

Morphazinamide is an anti-tuberculosis agent. Also, it is derived from Pyrazinamide (P840600), which is an anti-bacterial (tuberculostatic).

Definition

ChEBI: Morinamide is a member of pyrazines, a secondary carboxamide and a member of morpholines.

Manufacturing Process

98.5 parts by weight 2-pyrazinecarboxamide was mixed with 260 parts by volume of diethylamine. 91 parts by weight of 37% formaldehyde was added to above mixture by stirring for 30 minutes. The reaction mixture was spontaneously heated to 50°C. Then it heated to reflux for 5 hours on water bath. After that it was distilled to dryness at temperature between 40°-50°C. The residue was dissolved with about 200 parts by volume of ligroin (B.P. 60°C) by heating. The solution was filtered hot for removing the not reacted 2-pyrazinecarboxamide. Then it was cooled to -10°C and desired N- (diethylaminomethyl)-pyrazinecarboxylic acid amide discharged. It was filtered off and recrystallized from light petrol ester. Yield about 90%, MP: 47°-50°C.
500 parts by weight of N-(diethylaminomethyl)pyrazinecarboxylic acid amide and 2500 parts by volume of was mixed and heated by stirring to temperature 140°-150°C. At 60°-100°C a distillation begun and ended at 127°C (a boiling point of morpholine). The distillate consisted from diethylamine and morpholine. After 30-60 minutes the mixture was cooled to 50°C and distilled in vacuum to dryness. The residue was recrystallized from 400 parts by volume of benzene to give N-(morpholinomethyl)pyrazinecarboxamide, yield 92%, MP: 114°-117°C.

Therapeutic Function

Antitubercular

morinamide Preparation Products And Raw materials

Raw materials

Preparation Products

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morinamide Suppliers

Shaanxi DIDU pharmaceutical and Chemical Co., Ltd
Tel
15229059051
Email
1027@dideu.com
Country
China
ProdList
10011
Advantage
58
Shaanxi Didu New Materials Co. Ltd
Tel
+86-89586680 +86-13289823923
Email
1026@dideu.com
Country
China
ProdList
8670
Advantage
58

952-54-5, morinamideRelated Search:


  • morinamide
  • morphazinamide
  • B 2310
  • Morfazinamide
  • N-(Morpholinomethyl)-2-pyrazinecarboxamide
  • pyrazine-2-carboxylic acid morpholin-4-ylmethyl-amide
  • 2-Pyrazinecarboxamide, N-(4-morpholinylmethyl)-
  • 952-54-5