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CATHEPSIN G INHIBITOR I

Product Name
CATHEPSIN G INHIBITOR I
CAS No.
429676-93-7
Chemical Name
CATHEPSIN G INHIBITOR I
Synonyms
CATHEPSIN G INHIBITOR I;BOROXIN, TRIS(1-METHYLETHYL);Phosphonic acid, P-[2-[3-[[(1-benzoyl-4-piperidinyl)methylamino]carbonyl]-2-naphthalenyl]-1-(1-naphthalenyl)-2-oxoethyl]-
CBNumber
CB6310648
Molecular Formula
C36H33N2O6P
Formula Weight
620.64
MOL File
429676-93-7.mol
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CATHEPSIN G INHIBITOR I Property

Boiling point:
912.0±75.0 °C(Predicted)
Density 
1.40±0.1 g/cm3(Predicted)
storage temp. 
Store at -20°C
solubility 
Soluble in DMSO
pka
1.51±0.10(Predicted)
form 
Solid
Sensitive 
Light Sensitive
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Hazard and Precautionary Statements (GHS)

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N-Bromosuccinimide Price

Alfa Aesar
Product number
J65957
Product name
Cathepsin G Inhibitor I
Packaging
1mg
Price
$204
Updated
2023/06/20
Cayman Chemical
Product number
14928
Product name
Cathepsin G Inhibitor I
Purity
≥95%
Packaging
500μg
Price
$46
Updated
2024/03/01
Cayman Chemical
Product number
14928
Product name
Cathepsin G Inhibitor I
Purity
≥95%
Packaging
1mg
Price
$88
Updated
2024/03/01
Cayman Chemical
Product number
14928
Product name
Cathepsin G Inhibitor I
Purity
≥95%
Packaging
5mg
Price
$322
Updated
2024/03/01
TRC
Product number
C215205
Product name
Cathepsin G Inhibitor I
Packaging
5mg
Price
$445
Updated
2021/12/16
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CATHEPSIN G INHIBITOR I Chemical Properties,Usage,Production

Description

Cathepsin G inhibitor I is a potent and selective inhibitor of cathepsin G (IC50 = 53 nM). It weakly inhibits or has no effect on related proteases, including chymotrypsin, thrombin, plasmin, trypsin, tryptase, and elastase.

Uses

Cathepsin G inhibitor I is a potent and selective inhibitor of cathepsin G.

target

cathepsins G

References

[1] greco mn, hawkins mj, powell et, almond hr jr, corcoran tw, de garavilla l, kauffman ja, recacha r, chattopadhyay d, andrade-gordon p, maryanoff be. nonpeptide inhibitors of cathepsin g: optimization of a novel beta-ketophosphonic acid lead by structure-based drug design. j am chem soc. 2002;124(15):3810-1.

CATHEPSIN G INHIBITOR I Preparation Products And Raw materials

Raw materials

Preparation Products

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CATHEPSIN G INHIBITOR I Suppliers

429676-93-7, CATHEPSIN G INHIBITOR IRelated Search:


  • CATHEPSIN G INHIBITOR I
  • Phosphonic acid, P-[2-[3-[[(1-benzoyl-4-piperidinyl)methylamino]carbonyl]-2-naphthalenyl]-1-(1-naphthalenyl)-2-oxoethyl]-
  • BOROXIN, TRIS(1-METHYLETHYL)
  • 429676-93-7
  • C36H33N2O6P
  • A potent, selective, reversible, competitive, non-peptide inhibitor of cathepsin G.