GSK2807 Trifluoroacetate

Product Name: GSK2807 Trifluoroacetate
CAS No.: 2245255-66-5
Chemical Name: GSK2807 Trifluoroacetate
Synonyms: CS-2876;GSK2807 TFA;GSK2807 Trifluoroacetate;GSK2807,Inhibitor,GSK2807 Trifluoroacetate,inhibit,GSK-2807 Trifluoroacetate,Histone Methyltransferase,GSK 2807,GSK-2807;(S)-2-Amino-4-((((2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-dihydroxytetrahydrofuran-2-yl)methyl)(3-(dimethylamino)propyl)amino)butanoic acid 2,2,2-trifluoroacetic acid salt
CBNumber: CB64675587
Molecular Formula: C21H33F3N8O7
Formula Weight: 566.54
MOL File: 2245255-66-5.mol

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GSK2807 Trifluoroacetate Property

storage temp.: under inert gas (nitrogen or Argon) at 2–8 °C
solubility: DMSO:250.0(Max Conc. mg/mL);441.28(Max Conc. mM)
Water:50.0(Max Conc. mg/mL);88.26(Max Conc. mM)
form: Solid
color: White to yellow

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Hazard and Precautionary Statements (GHS)

Symbol(GHS)

Signal word

Warning

Hazard statements

H302Harmful if swallowed

H315Causes skin irritation

H319Causes serious eye irritation

H335May cause respiratory irritation

Precautionary statements

P261Avoid breathing dust/fume/gas/mist/vapours/spray.

P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

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N-Bromosuccinimide Price

ChemScene

Product number: CS-0046140
Product name: GSK2807Trifluoroacetate
Packaging: 5mg
Price: $250
Updated: 2021/12/16

AK Scientific

Product number: 8035EL
Product name: GSK2807Trifluoroacetate
Packaging: 5mg
Price: $276
Updated: 2021/12/16

ChemScene

Product number: CS-0046140
Product name: GSK2807Trifluoroacetate
Packaging: 10mg
Price: $350
Updated: 2021/12/16

ChemScene

Product number: CS-0046140
Product name: GSK2807Trifluoroacetate
Packaging: 25mg
Price: $750
Updated: 2021/12/16

AK Scientific

Product number: 8035EL
Product name: GSK2807Trifluoroacetate
Packaging: 100mg
Price: $1013
Updated: 2021/12/16

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GSK2807 Trifluoroacetate Chemical Properties,Usage,Production

Uses

GSK2807 Trifluoroacetate is a potent, selective and SAM-competitive inhibitor of SMYD3, with a Ki of 14 nM and an IC50 of 130 nM[1][2].

IC 50

SMYD3: 14 nM (Ki); SMYD3: 130 nM (IC₅₀)

References

[1] Van Aller GS, et al. Structure-Based Design of a Novel SMYD3 Inhibitor that Bridges the SAM-and MEKK2-Binding Pockets. Structure. 2016 May 3;24(5):774-781. DOI:10.1016/j.str.2016.03.010
[2] Kaniskan Hü, et al. Inhibitors of Protein Methyltransferases and Demethylases. Chem Rev. 2018 Feb 14;118(3):989-1068. DOI:10.1021/acs.chemrev.6b00801

GSK2807 Trifluoroacetate Preparation Products And Raw materials

Raw materials

Preparation Products

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GSK2807 Trifluoroacetate Suppliers

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2245255-66-5, GSK2807 TrifluoroacetateRelated Search:

GSK2807 Trifluoroacetate

CS-2876

(S)-2-Amino-4-((((2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-dihydroxytetrahydrofuran-2-yl)methyl)(3-(dimethylamino)propyl)amino)butanoic acid 2,2,2-trifluoroacetic acid salt

GSK2807 TFA

GSK2807,Inhibitor,GSK2807 Trifluoroacetate,inhibit,GSK-2807 Trifluoroacetate,Histone Methyltransferase,GSK 2807,GSK-2807

2245255-66-5