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MIN-101

Product Name
MIN-101
CAS No.
359625-79-9
Chemical Name
MIN-101
Synonyms
MT210;MT-210;MT 210;CYR-101;MIN-101;Roluperidone;CYR-101(Roluperidone);Roluperidone (MIN101);Roluperidone (CYR-101);Roluperidone, 10 mM in DMSO
CBNumber
CB73147776
Molecular Formula
C22H23FN2O2
Formula Weight
366.43
MOL File
359625-79-9.mol
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MIN-101 Property

storage temp. 
Store at -20°C
solubility 
DMSO:33.33(Max Conc. mg/mL);90.96(Max Conc. mM)
form 
A solid
color 
White to yellow
InChI
InChI=1S/C22H23FN2O2/c23-19-7-5-17(6-8-19)21(26)15-24-11-9-16(10-12-24)13-25-14-18-3-1-2-4-20(18)22(25)27/h1-8,16H,9-15H2
InChIKey
RNRYULFRLCBRQS-UHFFFAOYSA-N
SMILES
C1(=O)C2=C(C=CC=C2)CN1CC1CCN(CC(C2=CC=C(F)C=C2)=O)CC1
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Warning
Hazard statements

H303May be harmfulif swallowed

H320Causes eye irritation

Precautionary statements

P264Wash hands thoroughly after handling.

P264Wash skin thouroughly after handling.

P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

P312Call a POISON CENTER or doctor/physician if you feel unwell.

P337+P313IF eye irritation persists: Get medical advice/attention.

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N-Bromosuccinimide Price

Cayman Chemical
Product number
29773
Product name
CYR-101
Packaging
10mg
Price
$106
Updated
2024/03/01
Cayman Chemical
Product number
29773
Product name
CYR-101
Packaging
100mg
Price
$621
Updated
2024/03/01
Cayman Chemical
Product number
29773
Product name
CYR-101
Packaging
25mg
Price
$209
Updated
2024/03/01
Cayman Chemical
Product number
29773
Product name
CYR-101
Packaging
50mg
Price
$363
Updated
2024/03/01
ChemScene
Product number
CS-6971
Product name
Roluperidone
Purity
98.08%
Packaging
5mg
Price
$192
Updated
2021/12/16
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MIN-101 Chemical Properties,Usage,Production

Uses

Roluperidone (CYR-101) is a novel cyclic amide derivative that has high equipotent affinities for 5-HT2A and sigma-2 receptors (Ki of 7.53 nM and 8.19 nM for 5-HT2A and sigma-2, respectively).

IC 50

5-HT2A Receptor: 7.53 nM (Ki); Sigma-2 Receptor: 8.19 nM (Ki)

References

[1] Davidson M, et al. Efficacy and Safety of MIN-101: A 12-Week Randomized, Double-Blind, Placebo-Controlled Trial of a New Drug in Development for the Treatment of Negative Symptoms in Schizophrenia. Am J Psychiatry. 2017 Jul 28:appiajp201717010122. DOI:10.1176/appi.ajp.2017.17010122

MIN-101 Preparation Products And Raw materials

Raw materials

Preparation Products

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MIN-101 Suppliers

China 47 United States 6 Global 53
MedChemexpress LLC
Tel
021-58955995
Fax
609-228-5909
Email
sales@medchemexpress.cn
Country
United States
ProdList
4861
Advantage
58
TargetMol Chemicals Inc.
Tel
+1-781-999-5354; +17819995354
Email
marketing@targetmol.com
Country
United States
ProdList
32435
Advantage
58
InvivoChem
Tel
+1-708-310-1919 +1-13798911105
Fax
708-557-7486
Email
sales@invivochem.cn
Country
United States
ProdList
6391
Advantage
58
Aladdin Scientific
Tel
Email
tp@aladdinsci.com
Country
United States
ProdList
52923
Advantage
58
Cayman Chemical Company
Tel
--
Fax
--
Email
cayman@caymanchem.com
Country
United States
ProdList
6213
Advantage
81
MedChemExpress
Tel
--
Fax
--
Email
sales@medchemexpress.com
Country
United States
ProdList
6398
Advantage
58

359625-79-9, MIN-101Related Search:


  • MIN-101
  • CYR-101
  • Roluperidone (CYR-101)
  • MIN-101; MIN 101; MIN101; CYR-101; CYR 101; CYR101; MT-210; MT 210; MT210;
  • MT 210
  • MT210
  • MT-210
  • Roluperidone
  • 1H-Isoindol-1-one, 2-[[1-[2-(4-fluorophenyl)-2-oxoethyl]-4-piperidinyl]methyl]-2,3-dihydro-
  • CYR-101(Roluperidone)
  • MT210,MIN 101,5-hydroxytryptamine Receptor,CYR 101,MT 210,CYR101,Inhibitor,MIN101,inhibit,5-HT Receptor,Sigma Receptor,Roluperidone,Serotonin Receptor
  • Roluperidone (MIN101)
  • 2-((1-(2-(4-Fluorophenyl)-2-oxoethyl)piperidin-4-yl)methyl)isoindolin-1-one
  • Roluperidone, 10 mM in DMSO
  • 359625-79-9
  • APIS