Lobradimil

Product Name: Lobradimil
CAS No.: 159768-75-9
Chemical Name: Lobradimil
Synonyms: RMP 7;DRG0182;DRG 0182;DRG-0182;Lobradimil;ALK-01-040;Labradimil;Receptor-mediated permeabiliser-7;LabradiMil, LabrodiMil, RMP-7, LobradiMil;(Hyp3,b-(2-thienyl)-Ala5,Tyr(Me)8-()-Arg9)-Bradykinin
CBNumber: CB81309511
Molecular Formula: C49H75N15O12S
Formula Weight: 1098.29
MOL File: 159768-75-9.mol

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Lobradimil Property

Density: 1.53
pka: 2.34±0.24(Predicted)
form: Solid
color: White to off-white

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Hazard and Precautionary Statements (GHS)

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N-Bromosuccinimide Price

American Custom Chemicals Corporation

Product number: PEP0003686
Product name: LABRADIMIL
Purity: 95.00%
Packaging: 1MG
Price: $630.63
Updated: 2021/12/16

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Lobradimil Chemical Properties,Usage,Production

Uses

Adjuvant; receptor-mediated permeabiliser.

in vivo

Lobradimil (2.5-mg/kg bolus plus 10 mg/kg/h for 90 minutes) increases brain tumor permeability and shows hypotensive effects in RG2 glioma cells-implanted rats^[2].

Animal Model:	RG2 glioma cells-implanted rats^[2]
Dosage:	1.5-18 μg/kg
Administration:	i.v. infusion, 0.05 mL/min for 15min
Result:	Increased Carboplatin (HY-17393) uptake (up to 80%) into brain tumors in a dose-dependent manner.

IC 50

Bradykinin B2 Receptor (B2R): 0.54 nM (Ki)

Lobradimil Preparation Products And Raw materials

Raw materials

Preparation Products

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Lobradimil Suppliers

China 27 India 1 United States 5 Global 33

Shanghai Hanhong Scientific Co.,Ltd.

Tel: 021-54306202 13764082696
Email: info@hanhongsci.com
Country: China
ProdList: 42934
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Chemsky（shanghai）International Co.,Ltd.

Tel: 021-50135380
Email: shchemsky@163.com
Country: China
ProdList: 283
Advantage: 58

Chemsky (shanghai) International Co.,Ltd

Tel: 021-50135380
Email: shchemsky@sina.com
Country: China
ProdList: 15402
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BOC Sciences

Tel: 1-631-485-4226; 16314854226
Email: info@bocsci.com
Country: United States
ProdList: 12952
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Wuxi Zhongkun Biochemical Technology Co., Ltd.

Tel: 0510-85629785 18013409632
Fax: 051085625359
Email: sales@reading-chemicals.com
Country: China
ProdList: 15178
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Creative Peptides

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Email: info@creative-peptides.com
Country: United States
ProdList: 6083
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Hangzhou Peptidego Biotech Co.,Ltd.

Tel: 0571-87213919
Email: Eric@peptidego.com
Country: China
ProdList: 7408
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TargetMol Chemicals Inc.

Tel: +1-781-999-5354; +17819995354
Email: marketing@targetmol.com
Country: United States
ProdList: 32435
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Zhejiang J&C Biological Technology Co.,Limited

Tel: +1-2135480471
Email: sales@sarms4muscle.com
Country: China
ProdList: 10473
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Career Henan Chemica Co

Tel: +86-0371-86658258 +8613203830695
Fax: 0371-86658258
Email: laboratory@coreychem.com
Country: China
ProdList: 30229
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159768-75-9, LobradimilRelated Search:

Lobradimil

(Hyp3,β-(2-thienyl)-Ala5,Tyr(Me)8-(?)-Arg9)-Bradykinin Lobradimil

RMP 7

Lobradimil

(Hyp3,b-(2-thienyl)-Ala5,Tyr(Me)8-()-Arg9)-Bradykinin

H-Arg-Pro-Hyp-Gly-b-(2-thienyl)-Ala-Ser-Pro-Tyr(Me)-()-Arg-OH

LabradiMil, LabrodiMil, RMP-7, LobradiMil

(Hyp3,beta-(2-thienyl)-Ala5,Tyr(Me)8-(R)-Arg9)-Bradykinin

H-Arg-Pro-Hyp-Gly-b-(2-thienyl)-Ala-Ser-Pro-Tyr(Me)-psi(CH2NH)Arg-OH

(Hyp3,β-(2-thienyl)-Ala5,Tyr(Me)8-psi(CH2NH)Arg9)-Bradykinin

L-Arginine, L-arginyl-L-prolyl-(4R)-4-hydroxy-L-prolylglycyl-3-(2-thienyl)-L-alanyl-L-seryl-L-prolyl-O-methyl-L-tyrosyl-ψ(CH2-NH)-

(Hyp3,β-(2-thienyl)-Ala5,Tyr(Me)8-()-Arg9)-Bradykinin Lobradimil

(Hyp3,b-(2-thienyl)-Ala5,Tyr(Me)8-psi(CH2NH)Arg9)-Bradykinin (H-6578.0005)

ALK-01-040

DRG 0182

DRG0182

DRG-0182

Labradimil

Receptor-mediated permeabiliser-7

(Hyp3,β-(2-thienyl)-Ala?,Tyr(Me)?-psi(CH?NH)Arg?)-Bradykinin trifluoroacetate salt

(Hyp?,β-(2-thienyl)-Ala?,Tyr(Me)?-psi(CH?NH)Arg?)-Bradykinin

(Hyp3,β-(2-thienyl)-Ala5,Tyr(Me)8-(R)-Arg9)-Bradykinin

(Hyp 3,b-(2-thienyl)-Ala5,Tyr(Me)8-psi(CH2NH)Arg9)-Bradykinin trifluoroacetate salt

(Hyp3,β-(2-thienyl)-Ala5,Tyr(Me)8-psi(CH2NH)Arg9)-Bradykinin

159768-75-9