ChemicalBook > CAS DataBase List > N,N-DiMethyl-4-(4,4,5,5-tetraMethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole-1-ethanaMine

N,N-DiMethyl-4-(4,4,5,5-tetraMethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole-1-ethanaMine

Product Name
N,N-DiMethyl-4-(4,4,5,5-tetraMethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole-1-ethanaMine
CAS No.
877149-80-9
Chemical Name
N,N-DiMethyl-4-(4,4,5,5-tetraMethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole-1-ethanaMine
Synonyms
N,N-Dimethyl-2-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl);N,N-dimethyl-2-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-...;1-[2-(Dimethylamino)ethyl]-1H-pyrazole-4-boronic Acid Pinacol Ester;(1-(2-(dimethylamino)ethyl)-1H-pyrazol-4-yl)boronic acid pinacol ester;diMethyl({2-[4-(tetraMethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl]ethyl})aMine;N,N-DiMethyl-4-(4,4,5,5-tetraMethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole-1-ethanaMine;N,N-dimethyl-2-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazol-1-yl]ethanamine;1H-Pyrazole-1-ethanaMine, N,N-diMethyl-4-(4,4,5,5-tetraMethyl-1,3,2-dioxaborolan-2-yl)-;N,N-diMethyl-2-(4-(4,4,5,5-tetraMethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl)ethanaMine;N,N-dimethyl-2-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl)ethan-1-amine
CBNumber
CB82550288
Molecular Formula
C13H24BN3O2
Formula Weight
265.16
MOL File
877149-80-9.mol
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N,N-DiMethyl-4-(4,4,5,5-tetraMethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole-1-ethanaMine Property

Boiling point:
365.8±22.0 °C(Predicted)
Density 
1.04±0.1 g/cm3(Predicted)
storage temp. 
2-8°C
pka
8.93±0.28(Predicted)
Appearance
Colorless to light yellow Liquid
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
warning
Hazard statements

H302Harmful if swallowed

H315Causes skin irritation

H319Causes serious eye irritation

H335May cause respiratory irritation

Precautionary statements

P261Avoid breathing dust/fume/gas/mist/vapours/spray.

P264Wash hands thoroughly after handling.

P264Wash skin thouroughly after handling.

P270Do not eat, drink or smoke when using this product.

P271Use only outdoors or in a well-ventilated area.

P280Wear protective gloves/protective clothing/eye protection/face protection.

P301+P312IF SWALLOWED: call a POISON CENTER or doctor/physician IF you feel unwell.

P302+P352IF ON SKIN: wash with plenty of soap and water.

P304+P340IF INHALED: Remove victim to fresh air and Keep at rest in a position comfortable for breathing.

P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

P312Call a POISON CENTER or doctor/physician if you feel unwell.

P321Specific treatment (see … on this label).

P330Rinse mouth.

P332+P313IF SKIN irritation occurs: Get medical advice/attention.

P337+P313IF eye irritation persists: Get medical advice/attention.

P362Take off contaminated clothing and wash before reuse.

P403+P233Store in a well-ventilated place. Keep container tightly closed.

P405Store locked up.

P501Dispose of contents/container to..…

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N-Bromosuccinimide Price

AK Scientific
Product number
3944AC
Product name
N,N-Dimethyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole-1-ethanamine
Packaging
250mg
Price
$157
Updated
2021/12/16
ChemScene
Product number
CS-W000571
Product name
N,N-DIMETHYL-2-(4-(4,4,5,5-TETRAMETHYL-1,3,2-DIOXABOROLAN-2-YL)-1H-PYRAZOL-1-YL)ETHANAMINE
Packaging
1g
Price
$184
Updated
2021/12/16
SynQuest Laboratories
Product number
8H60-1-BL
Product name
Dimethyl({2-[4-(tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl]ethyl})amine
Purity
97.0%
Packaging
250mg
Price
$390
Updated
2021/12/16
ChemScene
Product number
CS-W000571
Product name
N,N-DIMETHYL-2-(4-(4,4,5,5-TETRAMETHYL-1,3,2-DIOXABOROLAN-2-YL)-1H-PYRAZOL-1-YL)ETHANAMINE
Packaging
100mg
Price
$58
Updated
2021/12/16
ChemScene
Product number
CS-W000571
Product name
N,N-DIMETHYL-2-(4-(4,4,5,5-TETRAMETHYL-1,3,2-DIOXABOROLAN-2-YL)-1H-PYRAZOL-1-YL)ETHANAMINE
Packaging
250mg
Price
$81
Updated
2021/12/16
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N,N-DiMethyl-4-(4,4,5,5-tetraMethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole-1-ethanaMine Chemical Properties,Usage,Production

Synthesis

269410-08-4

4584-46-7

877149-80-9

The reaction mixture was suspended in acetonitrile (30 mL) in the presence of cesium carbonate (6.72 g, 20.61 mmol) using 4-pyrazolylboronic acid pinacol ester (2 g, 10.31 mmol) and dimethylaminoethyl chloride hydrochloride (2.227 g, 15.46 mmol). The mixture was heated to reflux for 5 hours and then cooled to room temperature. The reaction solution was diluted with ether and filtered, and the filtrate was concentrated in vacuum to afford N,N-dimethyl-2-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl)ethanamine (2.61 g, 9.84 mmol, 95% yield) as an amber colored oil, which was used directly in the next step of the reaction.

References

[1] Patent: WO2011/54841, 2011, A1. Location in patent: Page/Page column 105
[2] Patent: US2014/45814, 2014, A1. Location in patent: Paragraph 0257; 0258
[3] Patent: WO2017/178416, 2017, A1. Location in patent: Page/Page column 116; 117
[4] Patent: WO2018/73602, 2018, A1. Location in patent: Page/Page column 99
[5] Patent: US2012/208798, 2012, A1. Location in patent: Page/Page column 47

N,N-DiMethyl-4-(4,4,5,5-tetraMethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole-1-ethanaMine Preparation Products And Raw materials

Raw materials

Preparation Products

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N,N-DiMethyl-4-(4,4,5,5-tetraMethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole-1-ethanaMine Suppliers

Shanghai Jian Chao Chemical Technology Co., Ltd.
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China
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Changzhou Chemscaler Pharmtech Co., Ltd.
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0519-81096292 15312577869
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chemscaler@yahoo.com.cn
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China
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Shanghai Raise Chemical Technology Co.,Ltd
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+86-021-50935922
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Shanghai Chainpharm Bio-medical Technology Co., Ltd.
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Changsha Luxing Bio-Chem Technology Co., Ltd.
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0731-88827538 15873153880
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Chengdu Aslee Biopharmaceuticals, Inc
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Nanjing Chalf-Pharm Technology Co., Ltd.
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Boron Technology (Beijing) Co., Ltd.
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View Lastest Price from N,N-DiMethyl-4-(4,4,5,5-tetraMethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole-1-ethanaMine manufacturers

Career Henan Chemical Co
Product
N,N-DiMethyl-4-(4,4,5,5-tetraMethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole-1-ethanaMine 877149-80-9
Price
US $1.00/KG
Min. Order
1KG
Purity
95%
Supply Ability
500KG
Release date
2018-08-19

877149-80-9, N,N-DiMethyl-4-(4,4,5,5-tetraMethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole-1-ethanaMineRelated Search:


  • N,N-DiMethyl-4-(4,4,5,5-tetraMethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole-1-ethanaMine
  • diMethyl({2-[4-(tetraMethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl]ethyl})aMine
  • N,N-diMethyl-2-(4-(4,4,5,5-tetraMethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl)ethanaMine
  • 1H-Pyrazole-1-ethanaMine, N,N-diMethyl-4-(4,4,5,5-tetraMethyl-1,3,2-dioxaborolan-2-yl)-
  • N,N-Dimethyl-2-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)
  • N,N-dimethyl-2-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazol-1-yl]ethanamine
  • N,N-dimethyl-2-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl)ethan-1-amine
  • 1-[2-(Dimethylamino)ethyl]-1H-pyrazole-4-boronic Acid Pinacol Ester
  • (1-(2-(dimethylamino)ethyl)-1H-pyrazol-4-yl)boronic acid pinacol ester
  • N,N-dimethyl-2-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-...
  • N,N-dimethyl-2-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl]ethanamine - [D11960]
  • 877149-80-9
  • C13H24BN3O2