H-P-CHLORO-PHE-D-CYS-BETA-(3-PYRIDYL)-ALA-D-TRP-N-ME-LYS-THR-CYS-2-NAL-NH2

Product Name: H-P-CHLORO-PHE-D-CYS-BETA-(3-PYRIDYL)-ALA-D-TRP-N-ME-LYS-THR-CYS-2-NAL-NH2
CAS No.: 341519-04-8
Chemical Name: H-P-CHLORO-PHE-D-CYS-BETA-(3-PYRIDYL)-ALA-D-TRP-N-ME-LYS-THR-CYS-2-NAL-NH2
Synonyms: PRL 3195;H-Phe(4-Cl)-D-Cys-β-(3-pyridyl)-Ala-D-Trp-N-Me-Lys-Thr-Cys-2-Nal-NH2;H-p-Chloro-Phe-D-Cys-β-(3-pyridyl)-Ala-D-Trp-N-Me-Lys-Thr-Cys-2-Nal-NH2;H-p-Chloro-Phe-D-Cys-b-(3-pyridyl)-Ala-D-Trp-N-Me-Lys-Thr-Cys-2-Nal-NH2;H-P-CHLORO-PHE-D-CYS-BETA-(3-PYRIDYL)-ALA-D-TRP-N-ME-LYS-THR-CYS-2-NAL-NH2;H-p-Chloro-Phe-D-Cys-β-(3-pyridyl)-Ala-D-Trp-N-Me-Lys-Thr-Cys-2-Nal-NH2 (Disulfide bond);H-P-CHLORO-PHE-D-CYS-BETA-(3-PYRIDYL)-ALA-D-TRP-N-ME-LYS-THR-CYS-2-NAL-NH2, (DISULFIDE BOND);H-p-Chloro-Phe-D-Cys-β-(3-pyridyl)-Ala-D-Trp-N-Me-Lys-Thr-Cys-2-Nal-NH(Disulfide bond) Trifluoroacetate salt;H-p-Chloro-Phe-D-Cys-β-(3-pyridyl)-Ala-D-Trp-N-Me-Lys-Thr-Cys-2-Nal-NH?(Disulfide bond) Trifluoroacetate salt;H-p-Chloro-Phe-D-Cys-b-(3-pyridyl)-Ala-D-Trp-N-Me-Lys-Thr-Cys-2-Nal-NH2 trifluoroacetate salt (Disulfide bond)
CBNumber: CB8277882
Molecular Formula: C58H69ClN12O9S2
Formula Weight: 1177.83
MOL File: 341519-04-8.mol

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H-P-CHLORO-PHE-D-CYS-BETA-(3-PYRIDYL)-ALA-D-TRP-N-ME-LYS-THR-CYS-2-NAL-NH2 Property

Boiling point:: 1522.8±65.0 °C(Predicted)
Density: 1.42±0.1 g/cm3(Predicted)
pka: 12.75±0.70(Predicted)
Sequence: {Phe<4Cl>}-{d-Cys}-{β-Ala<3-Py>}-{d-Trp}-{Lys}-Thr-Cys-{2-Nal}-NH2 (Disulfide bridge:Cys2-Cys7)

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Hazard and Precautionary Statements (GHS)

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N-Bromosuccinimide Price

Biosynth Carbosynth

Product number: FC109640
Product name: H-p-Chloro-Phe-D-Cys-b-(3-pyridyl)-Ala-D-Trp-N-Me-Lys-Thr-Cys-2-Nal-NH2 trifluoroacetate salt (Disulfide bond)
Packaging: 100ug
Price: $91
Updated: 2021/12/16

Biosynth Carbosynth

Product number: FC109640
Product name: H-p-Chloro-Phe-D-Cys-b-(3-pyridyl)-Ala-D-Trp-N-Me-Lys-Thr-Cys-2-Nal-NH2 trifluoroacetate salt (Disulfide bond)
Packaging: 250ug
Price: $180
Updated: 2021/12/16

Biosynth Carbosynth

Product number: FC109640
Product name: H-p-Chloro-Phe-D-Cys-b-(3-pyridyl)-Ala-D-Trp-N-Me-Lys-Thr-Cys-2-Nal-NH2 trifluoroacetate salt (Disulfide bond)
Packaging: 500ug
Price: $315
Updated: 2021/12/16

American Custom Chemicals Corporation

Product number: PEP0010270
Product name: H-P-CHLORO-PHE-D-CYS-BETA-(3-PYRIDYL)-ALA-D-TRP-N-ME-LYS-THR-CYS-2-NAL-NH2
Purity: 95.00%
Packaging: 5MG
Price: $505
Updated: 2021/12/16

Biosynth Carbosynth

Product number: FC109640
Product name: H-p-Chloro-Phe-D-Cys-b-(3-pyridyl)-Ala-D-Trp-N-Me-Lys-Thr-Cys-2-Nal-NH2 trifluoroacetate salt (Disulfide bond)
Packaging: 1mg
Price: $546
Updated: 2021/12/16

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H-P-CHLORO-PHE-D-CYS-BETA-(3-PYRIDYL)-ALA-D-TRP-N-ME-LYS-THR-CYS-2-NAL-NH2 Chemical Properties,Usage,Production

Uses

PRL 3195 is a somatostatin receptor antagonist with Kis of 6, 17, 66, 1000 and 1000 nM for human somatostatin receptors (sst5, sst2, sst3, sst1 and sst4, respectively)[1].

IC 50

hsst₅: 6 nM (Ki); hsst₂: 17 nM (Ki); hsst₃: 66 nM (Ki); hsst₁: 1000 nM (Ki); hsst₄: 1000 nM (Ki); rat urotensin II receptor: 429 nM (Ki); human urotensin II receptor: 1846 nM (Ki)

References

[1] Rossowski WJ, et al. Human urotensin II-induced aorta ring contractions are mediated by protein kinase C, tyrosine kinases and Rho-kinase: inhibition by somatostatin receptor antagonists. Eur J Pharmacol. 2002 Mar 8;438(3):159-70. DOI:10.1016/s0014-2999(02)01341-9

H-P-CHLORO-PHE-D-CYS-BETA-(3-PYRIDYL)-ALA-D-TRP-N-ME-LYS-THR-CYS-2-NAL-NH2 Preparation Products And Raw materials

Raw materials

Preparation Products

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H-P-CHLORO-PHE-D-CYS-BETA-(3-PYRIDYL)-ALA-D-TRP-N-ME-LYS-THR-CYS-2-NAL-NH2 Suppliers

China 32 Japan 1 United Kingdom 1 United States 3 Global 37

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341519-04-8, H-P-CHLORO-PHE-D-CYS-BETA-(3-PYRIDYL)-ALA-D-TRP-N-ME-LYS-THR-CYS-2-NAL-NH2Related Search:

H-P-CHLORO-PHE-D-CYS-BETA-(3-PYRIDYL)-ALA-D-TRP-N-ME-LYS-THR-CYS-2-NAL-NH2

H-p-Chloro-Phe-D-Cys-b-(3-pyridyl)-Ala-D-Trp-N-Me-Lys-Thr-Cys-2-Nal-NH2

H-p-Chloro-Phe-D-Cys-β-(3-pyridyl)-Ala-D-Trp-N-Me-Lys-Thr-Cys-2-Nal-NH(Disulfide bond) Trifluoroacetate salt

H-p-Chloro-Phe-D-Cys-β-(3-pyridyl)-Ala-D-Trp-N-Me-Lys-Thr-Cys-2-Nal-NH2 (Disulfide bond)

H-Phe(4-Cl)-D-Cys-β-(3-pyridyl)-Ala-D-Trp-N-Me-Lys-Thr-Cys-2-Nal-NH2

H-P-CHLORO-PHE-D-CYS-BETA-(3-PYRIDYL)-ALA-D-TRP-N-ME-LYS-THR-CYS-2-NAL-NH2

H-P-CHLORO-PHE-D-CYS-BETA-(3-PYRIDYL)-ALA-D-TRP-N-ME-LYS-THR-CYS-2-NAL-NH2, (DISULFIDE BOND)

H-p-Chloro-Phe-D-Cys-b-(3-pyridyl)-Ala-D-Trp-N-Me-Lys-Thr-Cys-2-Nal-NH2 trifluoroacetate salt (Disulfide bond)

L-Alaninamide, 4-chloro-L-phenylalanyl-D-cysteinyl-3-(3-pyridinyl)-L-alanyl-D-tryptophyl-N2-methyl-L-lysyl-L-threonyl-L-cysteinyl-3-(2-naphthalenyl)-, cyclic (2→7)-disulfide

PRL 3195

H-p-Chloro-Phe-D-Cys-β-(3-pyridyl)-Ala-D-Trp-N-Me-Lys-Thr-Cys-2-Nal-NH2

H-p-Chloro-Phe-D-Cys-β-(3-pyridyl)-Ala-D-Trp-N-Me-Lys-Thr-Cys-2-Nal-NH?(Disulfide bond) Trifluoroacetate salt

H-p-Chloro-Phe-D-Cys-β-(3-pyridyl)-Ala-D-Trp-N-Me-Lys-Thr-Cys-2-Nal-NH? trifluoroacetate salt (Disulfide bond)

341519-04-8

C58H69ClN12O9S2