ChemicalBook > CAS DataBase List > Kinase inhibitor-1
Kinase inhibitor-1
- Product Name
- Kinase inhibitor-1
- CAS No.
- 2135696-72-7
- Chemical Name
- Kinase inhibitor-1
- Synonyms
- Tarlox-TKI;Kinase inhibitor-1;TarloxTKI,Tarlox TKI;2-Butenamide, N-[4-[(3-bromo-4-chlorophenyl)amino]pyrido[3,4-d]pyrimidin-6-yl]-4-(dimethylamino)-, (2E)-
- CBNumber
- CB85419760
- Molecular Formula
- C19H18BrClN6O
- Formula Weight
- 461.74
- MOL File
- 2135696-72-7.mol
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Kinase inhibitor-1 Property
- Boiling point:
- 647.4±55.0 °C(Predicted)
- Density
- 1.552±0.06 g/cm3(Predicted)
- storage temp.
- Store at -20°C
- solubility
- DMSO: 100 mg/mL (216.57 mM); Water: < 0.1 mg/mL (insoluble)
- form
- Solid
- pka
- 9.68±0.43(Predicted)
- color
- Light yellow to yellow
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N-Bromosuccinimide Price
ChemScene
- Product number
- CS-0083039
- Product name
- Tarlox-TKI
- Purity
- 99.33%
- Packaging
- 5mg
- Price
- $450
- Updated
- 2021/12/16
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Kinase inhibitor-1 Chemical Properties,Usage,Production
Uses
Tarlox-TKI, the active metabolite of Tarloxotinib, is an irreversible pan-ErbB TKI (Tarlox-TKI)[1].
IC 50
EGFR
References
[1] Victoria Jackson-Patel, et al. Hypoxia tumour targeting with Tarloxotinib to improve clinical outcomes for patients with EGFR-dependent malignancies.
Kinase inhibitor-1 Preparation Products And Raw materials
Raw materials
Preparation Products
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Kinase inhibitor-1 Suppliers
- Tel
- +1-781-999-5354; +17819995354
- marketing@targetmol.com
- Country
- United States
- ProdList
- 32435
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- Tel
- +1-781-999-5354;
- support@targetmol.com
- Country
- United States
- ProdList
- 39035
- Advantage
- 58
- Tel
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- Fax
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- sales@medchemexpress.com
- Country
- United States
- ProdList
- 6398
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