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FLT3-IN-4

Product Name
FLT3-IN-4
CAS No.
2304799-09-3
Chemical Name
FLT3-IN-4
Synonyms
FLT3-IN-4;FLT3-IN-4, 10 mM in DMSO;1-{4-[4-amino-7-(prop-2-en-1-yl)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]phenyl}-3-(5-tert-butyl-1,2-oxazol-3-yl)urea;Urea, N-[4-[4-amino-7-(2-propen-1-yl)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]phenyl]-N'-[5-(1,1-dimethylethyl)-3-isoxazolyl]-
CBNumber
CB85540578
Molecular Formula
C23H25N7O2
Formula Weight
431.49
MOL File
2304799-09-3.mol
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FLT3-IN-4 Property

Boiling point:
589.1±50.0 °C(Predicted)
Density 
1.32±0.1 g/cm3(Predicted)
storage temp. 
Store at -20°C
solubility 
Soluble in DMSO
pka
12.68±0.70(Predicted)
form 
Solid
color 
White to off-white
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Hazard and Precautionary Statements (GHS)

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FLT3-IN-4 Chemical Properties,Usage,Production

Description

FLT3-IN-4 is a potent and orally effective Fms-like tyrosine receptor kinase 3 (FLT3; IC50=7 nM) inhibitor for treating acute myelogenous leukemia[1].

FLT3-IN-4 (Compound 9u) shows potent inhibitory activities against MV4-11 and Molm-13 cells with IC50 values are 0.089±0.001 nM and 0.022±0.003 nM, respectively[1].

References

[1]. Yuan X, et al. Identification of Pyrrolo[2,3- d]pyrimidine-Based Derivatives as Potent and Orally Effective Fms-like Tyrosine Receptor Kinase 3 (FLT3) Inhibitors for Treating Acute Myelogenous Leukemia. J Med Chem. 2019 Apr 25;62(8):4158-4173.

FLT3-IN-4 Preparation Products And Raw materials

Raw materials

Preparation Products

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FLT3-IN-4 Suppliers

TargetMol Chemicals Inc.
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Aladdin Scientific
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2304799-09-3, FLT3-IN-4Related Search:


  • FLT3-IN-4
  • Urea, N-[4-[4-amino-7-(2-propen-1-yl)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]phenyl]-N'-[5-(1,1-dimethylethyl)-3-isoxazolyl]-
  • 1-{4-[4-amino-7-(prop-2-en-1-yl)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]phenyl}-3-(5-tert-butyl-1,2-oxazol-3-yl)urea
  • FLT3-IN-4, 10 mM in DMSO
  • 2304799-09-3