ChemicalBook > CAS DataBase List > Abarelix (acetate)
Abarelix (acetate)
- Product Name
- Abarelix (acetate)
- CAS No.
- 785804-17-3
- Chemical Name
- Abarelix (acetate)
- Synonyms
- N-acetyl-3-(2-naphthalenyl)-D-alanyl-4-chloro-D-phenylalanyl-3-(3-pyridinyl)-D-alanyl-L-seryl-N-methyl-L-tyrosyl-D-asparaginyl-L-leucyl-N6-(1-methylethyl)-L-lysyl-L-prolyl-D-alaninamide, acetate salt
- CBNumber
- CB85540952
- Molecular Formula
- C74H99ClN14O16
- Formula Weight
- 1476.14
- MOL File
- 785804-17-3.mol
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Abarelix (acetate) Property
- storage temp.
- Store at -20°C
- solubility
- DMF: 30 mg/ml; DMSO: 30 mg/ml; Ethanol: 30 mg/ml; PBS (pH 7.2): 5 mg/ml
- form
- A crystalline solid
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N-Bromosuccinimide Price
Cayman Chemical
- Product number
- 28746
- Product name
- Abarelix (acetate)
- Packaging
- 1mg
- Price
- $25
- Updated
- 2024/03/01
Cayman Chemical
- Product number
- 28746
- Product name
- Abarelix (acetate)
- Packaging
- 25mg
- Price
- $281
- Updated
- 2024/03/01
Cayman Chemical
- Product number
- 28746
- Product name
- Abarelix (acetate)
- Packaging
- 5mg
- Price
- $69
- Updated
- 2024/03/01
Cayman Chemical
- Product number
- 28746
- Product name
- Abarelix (acetate)
- Packaging
- 10mg
- Price
- $125
- Updated
- 2024/03/01
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Abarelix (acetate) Chemical Properties,Usage,Production
Description
Abarelix acetate is a synthetic third generation gonadotropin-releasing hormone receptor (GnRHR) antagonist. It increases histamine release from rat peritoneal mast cells in vitro and from a human skin model ex vivo. In vivo, abarelix decreases plasma luteinizing hormone (LH) levels six hours post-treatment in castrated rats, with levels returning to baseline within 24 hours.3 Abarelix (2 mg/kg) also transiently decreases plasma testosterone levels in intact rats, with levels returning to baseline within seven days post-treatment. Formulations containing abarelix have previously been used in the treatment of advanced prostate cancer.
Abarelix (acetate) Preparation Products And Raw materials
Raw materials
Preparation Products
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Abarelix (acetate) Suppliers
- Tel
- --
- Fax
- --
- cayman@caymanchem.com
- Country
- United States
- ProdList
- 6213
- Advantage
- 81