methoctramine tetrahydrochloride hemihydrate

Product Name
methoctramine tetrahydrochloride hemihydrate
CAS No.
104807-46-7
Chemical Name
methoctramine tetrahydrochloride hemihydrate
Synonyms
methoctramine;MethoctraMine hydrate;methoctramine hemihydrate;Methoctramine tetrahydrochloride hydrate;methoctramine tetrahydrochloride hemihydrate;N,N′-bis[6-[[(2-Methoxyphenyl)methyl]amino]hexyl]-1,8-octane diamine tetrahydrochloride hydrate;Methoctramine hemihydrate tetrahydrochloride, N,Nμ-bis[6-[[(2-Methoxyphenyl)methyl]amino]hexyl]-1,8-octane diamine hemihydrate tetrahydrochloride
CBNumber
CB91216157
Molecular Formula
2C36H62N4O2.4ClH.H2O
Formula Weight
1329.68
MOL File
104807-46-7.mol
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methoctramine tetrahydrochloride hemihydrate Property

storage temp. 
2-8°C
solubility 
H2O: >20mg/mL
form 
solid
color 
white
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Safety

WGK Germany 
3
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Hazard and Precautionary Statements (GHS)

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N-Bromosuccinimide Price

Sigma-Aldrich
Product number
M105
Product name
Methoctramine hydrate
Purity
≥97% (NMR), solid
Packaging
10mg
Price
$223
Updated
2024/03/01
Sigma-Aldrich
Product number
M105
Product name
Methoctramine hydrate
Purity
≥97% (NMR), solid
Packaging
25mg
Price
$444
Updated
2024/03/01
Cayman Chemical
Product number
24317
Product name
Methoctramine
Purity
≥95%
Packaging
5mg
Price
$116
Updated
2024/03/01
Cayman Chemical
Product number
24317
Product name
Methoctramine
Purity
≥95%
Packaging
10mg
Price
$208
Updated
2024/03/01
Sigma-Aldrich
Product number
M105
Product name
Methoctramine hydrate
Purity
≥97% (NMR), solid
Packaging
100mg
Price
$1510
Updated
2024/03/01
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methoctramine tetrahydrochloride hemihydrate Chemical Properties,Usage,Production

Uses

Methoctramine is a muscarinic M2 receptor antagonist.

Uses

Methoctramine hydrate has been used:

  • As a muscarinic receptor 2 antogonist.
  • As a test molecule to check its effect on premature osteogenic differentiation of HGPS (Hutchinson-Gilford progeria syndrome) iPS (induced pluripotent)-derived mesenchymal stem cells.

Definition

ChEBI: A hydrochloride obtained by combining methoctramine with four molar equivalents of hydrochloric acid.

General Description

Methoctramine (N, N′-bis [6-[[(2-methoxyphenyl)-methyl] hexyl]-1, 8-octane] diamine) is a derivative of polymethylene tetramine.

Biochem/physiol Actions

Methoctramine is a selective M2 muscarinic receptor antagonist at nM concentrations. At mM concentrations, methoctramine directly inhibits the high affinity GTPase activity of G proteins. In oesophageal muscle, acetylcholine-mediated increase in calcium and arachidonic acid release were reduced by the M2 receptor antagonist, methoctramine. Methoctramine infused bilaterally in the dorsolateral striatum, considerably enhanced memory in cognitively impaired aged rats. Methoctramine plays a vital role in muscarinic receptor classification.

methoctramine tetrahydrochloride hemihydrate Preparation Products And Raw materials

Raw materials

Preparation Products

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methoctramine tetrahydrochloride hemihydrate Suppliers

Sigma-Aldrich
Tel
021-61415566 800-8193336
Email
orderCN@merckgroup.com
Country
China
ProdList
51456
Advantage
80
ChemeGen(Shanghai) Biotechnology Co.,Ltd.
Tel
18818260767
Fax
QQ 3610331285
Email
sales@chemegen.com
Country
China
ProdList
11217
Advantage
58
Energy Chemical
Tel
021-58432009 400-005-6266
Fax
021-58436166
Email
marketing1@energy-chemical.com
Country
China
ProdList
44808
Advantage
58
MedBioPharmaceutical Technology Inc
Tel
021-69568360 18916172912
Email
order@med-bio.cn
Country
China
ProdList
8140
Advantage
58
Shanghai Universal Biotech Co.,Ltd
Tel
15921930842 15921930842
Email
zhouzz@univ-bio.com
Country
China
ProdList
24990
Advantage
58
Jiangsu Aikon Biopharmaceutical R&D Co.,Ltd
Tel
13915962545
Email
2881759498@qq.com
Country
China
ProdList
2016
Advantage
58
Hangzhou MolCore BioPharmatech Co.,Ltd.
Tel
+86-057181025280; +8617767106207
Fax
0571-85806285
Email
sales@molcore.com
Country
China
ProdList
49734
Advantage
58
Guangzhou WeiBo Chemical Co., Ltd.
Tel
--
Fax
--
Email
weibochem@163.com
Country
China
ProdList
6187
Advantage
67

104807-46-7, methoctramine tetrahydrochloride hemihydrateRelated Search:


  • methoctramine hemihydrate
  • methoctramine tetrahydrochloride hemihydrate
  • methoctramine
  • Methoctramine hemihydrate tetrahydrochloride, N,Nμ-bis[6-[[(2-Methoxyphenyl)methyl]amino]hexyl]-1,8-octane diamine hemihydrate tetrahydrochloride
  • Methoctramine tetrahydrochloride hydrate
  • N,N′-bis[6-[[(2-Methoxyphenyl)methyl]amino]hexyl]-1,8-octane diamine tetrahydrochloride hydrate
  • MethoctraMine hydrate
  • 104807-46-7
  • C36H62N4O24HCl05H2O
  • C36H66Cl4N4O2