ChemicalBook > CAS DataBase List > SUVN-502
SUVN-502
- Product Name
- SUVN-502
- CAS No.
- 1791396-46-7
- Chemical Name
- SUVN-502
- Synonyms
- SUVN-502;SUVN-502 mesylate;SUVN-502 dimesylate;Masupirdine mesylate;Masupirdine mesylate, 10 mM in DMSO
- CBNumber
- CB93364117
- Molecular Formula
- C22H28BrN3O6S2
- Formula Weight
- 574.51
- MOL File
- 1791396-46-7.mol
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SUVN-502 Property
- storage temp.
- Store at -20°C
- solubility
- Soluble in DMSO
- form
- Solid
- color
- Pale purple to purple
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N-Bromosuccinimide Price
ChemScene
- Product number
- CS-0087572
- Product name
- Masupirdinemesylate
- Purity
- 99.58%
- Packaging
- 1mg
- Price
- $150
- Updated
- 2021/12/16
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SUVN-502 Chemical Properties,Usage,Production
Uses
Masupirdine mesylate (SUVN-502 mesylate) is a potent, selective, orally bioavailable, and brain penetrant 5-HT6 receptor antagonist (Ki of 2.04 nM for human 5-HT6 receptor). Masupirdine mesylate (SUVN-502 mesylate) shows high selectivity over 5-HT2A receptor and other 100 target sites, and has potential for treatment of Alzheimer's disease[1].
IC 50
5-HT6 Receptor: 2.04 nM (Ki)
References
[1] Nirogi R, et al. Discovery and Development of 1-[(2-Bromophenyl)sulfonyl]-5-methoxy-3-[(4-methyl-1-piperazinyl)methyl]-1H-indole Dimesylate Monohydrate (SUVN-502): A Novel, Potent, Selective and Orally Active Serotonin 6 (5-HT6) Receptor Antagonist for Po DOI:10.1021/acs.jmedchem.6b01662
SUVN-502 Preparation Products And Raw materials
Raw materials
Preparation Products
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SUVN-502 Suppliers
- Tel
- +1-781-999-5354; +17819995354
- marketing@targetmol.com
- Country
- United States
- ProdList
- 32435
- Advantage
- 58
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- Fax
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- sales@medchemexpress.com
- Country
- United States
- ProdList
- 6398
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