PSB CB5

Product Name: PSB CB5
CAS No.: 1627710-30-8
Chemical Name: PSB CB5
Synonyms: PSB CB5;GPR18IN32;GPR18-IN-32;GPR18 IN 32;CID-85469571;CID-85469571|||GPR18-IN-32;5H-Imidazo[2,1-b][1,3]thiazin-3(2H)-one, 2-[[3-[(4-chlorophenyl)methoxy]phenyl]methylene]-6,7-dihydro-, (2Z)-
CBNumber: CB98202883
Molecular Formula: C20H17ClN2O2S
Formula Weight: 384.88
MOL File: 1627710-30-8.mol

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PSB CB5 Property

Boiling point:: 549.9±60.0 °C(Predicted)
Density: 1.35±0.1 g/cm3(Predicted)
storage temp.: -20°C
solubility: Soluble in DMSO (up to 25 mg/ml)
pka: -1.84±0.20(Predicted)
form: solid
color: Pale yellow
Stability:: Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.

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Hazard and Precautionary Statements (GHS)

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N-Bromosuccinimide Price

Tocris

Product number: 6372
Product name: PSBCB5
Purity: ≥98%(HPLC)
Packaging: 50
Price: $873
Updated: 2021/12/16

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PSB CB5 Chemical Properties,Usage,Production

Description

PSB-CB5 (1627710-30-8) is a potent and selective GPR18 antagonist (IC50?= 0.279 μM) exhibiting >36-fold selectivity against GPR55 and CB1 and 14-fold selectivity against CB2.1? Inhibits N-arachidonylglycine-induced acrosomal exocytosis in human spermatozoa indicating that GPR18 may be involved in physiological processes of human spermatozoa.2

storage

Store at -20°C

References

1) Rempel?et al. (2014),?Bicyclic imidazole-4-one derivatives: a new class of antagonists for the orphan G protein-coupled receptors GPR18 and GPR55; Med. Chem. Comm., 5?632 2) Flegel?et al.?(2016),?Characterization of Non-Olfactory GPCRs in Human Sperm With a Focus on GPR18; Sci. Rep.,?6?32255

PSB CB5 Preparation Products And Raw materials

Raw materials

Preparation Products

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PSB CB5 Suppliers

China 10 United States 4 Global 14

Shanghai EFE Biological Technology Co., Ltd.

Tel: 021-65675885 18964387627
Fax: 021-65675885
Email: info@efebio.com
Country: China
ProdList: 9804
Advantage: 58

Tianjin Kailiqi Biotechnology Co., Ltd.

Tel: 15076683720
Fax: 022-23754520
Email: klq@cw-bio.com
Country: China
ProdList: 5960
Advantage: 55

Shanghai Changyu Medical Technology Co. Ltd.

Tel: +86-13301875428
Email: sales@changyuhe.com
Country: China
ProdList: 311
Advantage: 58

Shanghai Hongye Biotechnology Co. Ltd

Tel: 400-9205774
Email: sales@glpbio.cn
Country: China
ProdList: 6777
Advantage: 58

TargetMol Chemicals Inc.

Tel: +1-781-999-5354 +1-00000000000
Email: marketing@targetmol.com
Country: United States
ProdList: 32161
Advantage: 58

Changzhou Furuisi Biotechnology Co., Ltd

Tel: 0519-85524369
Email: 3477467573@qq.com
Country: China
ProdList: 8617
Advantage: 58

Nantong Hi-Future Biotechnology Co., Ltd

Tel: 18051384581
Email: sales@chemhifuture.com
Country: China
ProdList: 3021
Advantage: 58

TargetMol Chemicals Inc.

Tel: 4008200310
Email: marketing@tsbiochem.com
Country: China
ProdList: 24644
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R&D Systems, Inc

Tel: 18003437475
Fax: 1-612-656-4400
Email: rdname@qq.com
Country: China
ProdList: 35733
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Aladdin Scientific

Tel
Email: tp@aladdinsci.com
Country: United States
ProdList: 52924
Advantage: 58

1627710-30-8, PSB CB5Related Search:

SR 144528 CYCLOPAMINE Nalmefene hydrochloride

PSB CB5

CID-85469571

GPR18 IN 32

GPR18IN32

GPR18-IN-32

5H-Imidazo[2,1-b][1,3]thiazin-3(2H)-one, 2-[[3-[(4-chlorophenyl)methoxy]phenyl]methylene]-6,7-dihydro-, (2Z)-

CID-85469571|||GPR18-IN-32

1627710-30-8