(S)-5-IODO-3-[(2-AZETIDINYL)-METHOXY]PYRIDINE
(S)-5-IODO-3-[(2-AZETIDINYL)-METHOXY]PYRIDINE Basic information
- Product Name:
- (S)-5-IODO-3-[(2-AZETIDINYL)-METHOXY]PYRIDINE
- Synonyms:
-
- PYRIDINE, 3-[(2S)-2-AZETIDINYLMETHOXY]-5-IODO-,TRIFLUOROACETATE
- (S)-5-IODO-3-[(2-AZETIDINYL)-METHOXY]PYRIDINE
- 5-IODO-ALPHA-85380 DIHYDROCHLORIDE
- 3-[(2S)-2-AZETIDINYLMETHOXY]-5-IODOPYRIDINE DIHYDROCHLORIDE
- 3-[(2S)-2-AZETIDINYLMETHOXY]-5-IODO-PYRIDINE TRIFLUOROACETATE
- IAP TFA
- IAP TRIFLUOROACETATE
- 5-Iodo-A-853802HCl
- CAS:
- 213764-92-2
- MF:
- C28H27F15I2N4O12
- MW:
- 1150.32
- Mol File:
- 213764-92-2.mol
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(S)-5-IODO-3-[(2-AZETIDINYL)-METHOXY]PYRIDINE Chemical Properties
- storage temp.
- Desiccate at +4°C
- CAS DataBase Reference
- 213764-92-2
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(S)-5-IODO-3-[(2-AZETIDINYL)-METHOXY]PYRIDINE Usage And Synthesis
Chemical Properties
Colourless oil
Uses
5-IODO-A-85380 Dihydrochloride is a highly potent and subtype-selective agonist for AChR α4β2 and AChR α6β2.
Biological Activity
A highly potent and subtype-selective agonist for the α 4 β 2 and α 6 β 2 nicotinic acetylcholine receptors. Activates α -CTx-MII-sensitive and -insensitive components of [ 3 H]dopamine release from rat striatal synaptosomes, corresponding to α 6 β 2 and α 4 β 2 (EC 50 values are 12.7 and ~35 nM respectively). ~5000- , 25000- and 140000-fold selective over α 3 β 4, α 7 and muscle nAChR receptors respectively.
(S)-5-IODO-3-[(2-AZETIDINYL)-METHOXY]PYRIDINESupplier
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