Basic information Safety Supplier Related

MMP INHIBITOR I

Basic information Safety Supplier Related

MMP INHIBITOR I Basic information

Product Name:
MMP INHIBITOR I
Synonyms:
  • P-aminobenzoyl-gly-pro-D-leu-D-ala*hydroxamic aci
  • 4-ABZ-GLY-PRO-D-LEU-D-ALA-NHOH
  • METALLOPROTEASE INHIBITOR 1
  • MATRIX METALLOPROTEINASE INHIBITOR I
  • 4-aminobenzoyl-gly-pro-d-leu-d-ala hydroxamic acid
  • D-AlaninaMide, N-(4-aMinobenzoyl)glycyl-L-prolyl-D-leucyl-N-hydroxy-
  • 4-Abz-Gly-Pro-D-Leu-D-Ala-NHOH trifluoroacetate salt
  • H-4-ABZ-GLY-PRO-D-LEU-D-ALA-NHOH
CAS:
124168-73-6
MF:
C23H34N6O6
MW:
490.55
Product Categories:
  • Inhibitor of human matrix metalloproteinases.
Mol File:
124168-73-6.mol
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MMP INHIBITOR I Chemical Properties

Density 
1.288±0.06 g/cm3(Predicted)
storage temp. 
-20°C
solubility 
H2O: 1 mg/mL
pka
9.34±0.40(Predicted)
form 
solid
color 
white
Water Solubility 
water: 1mg/mL
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Safety Information

WGK Germany 
3

MSDS

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MMP INHIBITOR I Usage And Synthesis

Uses

FN-439 is a selective collagenase-1 inhibitor. FN-439 inhibits collagenase-1 with an IC50 value of 1 μM. FN-439 can be used for the research of cancer and inflammation[1][2].

Biological Activity

Collagenase Inhibitor

in vivo

FN-439 significantly decreases neutrophils and macrophages, shows extensive bone formation and active cementogenesis in the periapical region when has a combination with ofloxaci[2].

References

[1] U Benbow, et al. Human breast cancer cells activate procollagenase-1 and invade type I collagen: invasion is inhibited by all-trans retinoic acid. Clin Exp Metastasis. 1999 May;17(3):231-8. DOI:10.1023/a:1006639214618
[2] H Anan, et al. Effects of a combination of an antibacterial agent (ofloxacin) and a collagenase inhibitor (FN-439) on the healing of rat periapical lesions. J Endod. 1996 Dec;22(12):668-73. DOI:10.1016/S0099-2399(96)80061-6

MMP INHIBITOR ISupplier

3B Pharmachem (Wuhan) International Co.,Ltd.
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GL Biochem (Shanghai) Ltd
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VDM Biochemicals
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Shanghai Hanhong Scientific Co.,Ltd.
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Chemsky (shanghai) International Co.,Ltd
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