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5-Bromo-6-chloro-n-(4-(chlorodifluoromethoxy)phenyl)nicotinamide

Basic information Safety Supplier Related

5-Bromo-6-chloro-n-(4-(chlorodifluoromethoxy)phenyl)nicotinamide Basic information

Product Name:
5-Bromo-6-chloro-n-(4-(chlorodifluoromethoxy)phenyl)nicotinamide
Synonyms:
  • 3-Pyridinecarboxamide, 5-bromo-6-chloro-N-[4-(chlorodifluoromethoxy)phenyl]-
  • 5-bromo-6-chloro-N-(4-(chlorodifluoromethoxy)phenyl)pyridine-3-carboxamide
  • 5-bromo-6-chloro-N-(4-(chlorodifluoromethoxy)phenyl)nicotinamide
CAS:
1491150-22-1
MF:
C13H7BrCl2F2N2O2
MW:
412.01
Mol File:
1491150-22-1.mol
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5-Bromo-6-chloro-n-(4-(chlorodifluoromethoxy)phenyl)nicotinamide Chemical Properties

Boiling point:
399.0±42.0 °C(Predicted)
Density 
1.745±0.06 g/cm3(Predicted)
pka
10.00±0.70(Predicted)
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5-Bromo-6-chloro-n-(4-(chlorodifluoromethoxy)phenyl)nicotinamide Usage And Synthesis

Uses

5-Bromo-6-chloro-n-(4-(chlorodifluoromethoxy)phenyl)nicotinamide is a pharmaceutical intermediate compound used in the preparation of the anti-tumour drug Asciminib. Asciminib is a tyrosine kinase inhibitor (TKI) indicated for the treatment of chronic phase Philadelphia chromosome-positive chronic myeloid leukaemia (Ph+ CML).

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