ISAMOLTANE HEMIFUMARATE
ISAMOLTANE HEMIFUMARATE Basic information
- Product Name:
- ISAMOLTANE HEMIFUMARATE
- Synonyms:
-
- 1-[(1-Methylethyl)amino]-3-[2-(1H-pyrrol-1-yl)phenoxy]propan-2-ol fumarate (2:1) salt
- 1-[(1-Methylethyl)amino]-3-[2-(1H-pyrrol-1-yl)phenoxy]-2-propanol
- CG-361A
- 2-Propanol, 1-((1-methylethyl)amino)-3-(2-(1H-pyrrol-1-yl)phenoxy)-
- Isamoltanum
- Isamoltanum [latin]
- 1-((1-Methylethyl)amino)-3-(2-((1H)-pyrrol-1-yl))propan-2-olhemifumarate
- 1-(2-(1H-Pyrrol-1-yl)phenoxy)-3-(isopropylamino)propan-2-ol hemifumarate
- CAS:
- 55050-95-8
- MF:
- C16H22N2O2
- MW:
- 274.36
- Product Categories:
-
- Serotonin receptor
- Mol File:
- 55050-95-8.mol
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ISAMOLTANE HEMIFUMARATE Chemical Properties
- Boiling point:
- 443.4±40.0 °C(Predicted)
- Density
- 1.09±0.1 g/cm3(Predicted)
- storage temp.
- Desiccate at +4°C
- pka
- 13.76±0.20(Predicted)
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ISAMOLTANE HEMIFUMARATE Usage And Synthesis
Uses
Isamoltane hemifumarate is a selective SR-1B antagonist.
Definition
ChEBI: 1-(propan-2-ylamino)-3-[2-(1-pyrrolyl)phenoxy]-2-propanol is a member of pyrroles.
Biological Activity
5-HT 1B antagonist, approximately 30-fold selective over 5-HT 1A . Also possesses affinity for β -adrenergic receptors.