BOC-ALA-ALA-D-TRP-PHE-D-PRO-PRO-NLE-NH2
BOC-ALA-ALA-D-TRP-PHE-D-PRO-PRO-NLE-NH2 Basic information
- Product Name:
- BOC-ALA-ALA-D-TRP-PHE-D-PRO-PRO-NLE-NH2
- Synonyms:
-
- BOC-ALA-ALA-D-TRP-PHE-D-PRO-PRO-NLE-NH2
- GR 87389
- L-Norleucinamide, N-[(1,1-dimethylethoxy)carbonyl]-L-alanyl-L-alanyl-D-tryptophyl-L-phenylalanyl-D-prolyl-L-prolyl- (9CI)
- L-Norleucinamide,N-[(1,1-dimethylethoxy)carbonyl]-L-alanyl-L-alanyl-D-tryptophyl-L-phenylalanyl-D-prolyl-L-prolyl-
- CAS:
- 141663-86-7
- MF:
- C47H65N9O9
- MW:
- 900.07
- Mol File:
- 141663-86-7.mol
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BOC-ALA-ALA-D-TRP-PHE-D-PRO-PRO-NLE-NH2 Chemical Properties
- storage temp.
- -15°C
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BOC-ALA-ALA-D-TRP-PHE-D-PRO-PRO-NLE-NH2 Usage And Synthesis
Uses
GR 87389 is a potent NK2 receptor antagonist. GR 87389 antagonized GA 64349-induced smooth muscle strips contractions in a competitive manner in the human detrusor, prostate and prostatic urethra[1][2].
IC 50
NK2
References
[1] Saffroy M, et, al. Presence of NK2 binding sites in the rat brain. J Neurochem. 2001 Dec;79(5):985-96. DOI:10.1046/j.1471-4159.2001.00633.x
[2] Palea S, et, al. Pharmacological characterization of tachykinin NK2 receptors on isolated human urinary bladder, prostatic urethra and prostate. J Pharmacol Exp Ther. 1996 May;277(2):700-5. PMID:8627548
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