ChemicalBook > Product Catalog > Biologics > Biochemical Reagents > Antagonist > 4-DIMETHYLAMINO-7-(4-ETHYL-PHENYL)-7H-9-THIA-1,5,7-TRIAZA-FLUOREN-8-ONE
4-DIMETHYLAMINO-7-(4-ETHYL-PHENYL)-7H-9-THIA-1,5,7-TRIAZA-FLUOREN-8-ONE
4-DIMETHYLAMINO-7-(4-ETHYL-PHENYL)-7H-9-THIA-1,5,7-TRIAZA-FLUOREN-8-ONE Basic information
- Product Name:
- 4-DIMETHYLAMINO-7-(4-ETHYL-PHENYL)-7H-9-THIA-1,5,7-TRIAZA-FLUOREN-8-ONE
- Synonyms:
-
- 4-DIMETHYLAMINO-7-(4-ETHYL-PHENYL)-7H-9-THIA-1,5,7-TRIAZA-FLUOREN-8-ONE
- Pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-4(3H)-one, 9-(dimethylamino)-3-(4-ethylphenyl)-
- A-794282
- A 794282,A794282
- 9-(Dimethylamino)-3-(4-ethylphenyl)pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-4(3H)-one
- CAS:
- 869802-44-8
- MF:
- C19H18N4OS
- MW:
- 350.44
- Mol File:
- 869802-44-8.mol
More
Less
4-DIMETHYLAMINO-7-(4-ETHYL-PHENYL)-7H-9-THIA-1,5,7-TRIAZA-FLUOREN-8-ONE Usage And Synthesis
Description
A-794282 is a selective mGluR1 antagonist.
Uses
A-794282 is a compound with analgesic activity and is a selective mGlu1 receptor antagonist that significantly reduces pain behaviors in a postoperative pain model, but motor side effects may occur at higher doses.
IC 50
mGluR1
References
[1] Analgesic activity of metabotropic glutamate receptor 1 antagonists on spontaneous post-operative pain in rats DOI:10.1016/j.ejphar.2007.09.047
[2] [Research progress of selective mGluR1 antagonists] PMID:22242445
4-DIMETHYLAMINO-7-(4-ETHYL-PHENYL)-7H-9-THIA-1,5,7-TRIAZA-FLUOREN-8-ONESupplier
Ningbo Chaoming Biotechnology Co., Ltd Gold
- Tel
- 13301662590
- mandy@atkchemical.com
Shanghai YuanYe Biotechnology Co., Ltd.
- Tel
- 021-61312847; 18021002903
- 3008007409@qq.com
TargetMol Chemicals Inc.
- Tel
- +1-781-999-5354; +17819995354
- marketing@targetmol.com
ShangHai ChuanQian Chemcial Technique Centre
- Tel
- 15869524721
- 3525679403@qq.com
cjbscvictory
- Tel
- 13348960310
- 3003867561@qq.com