ChemicalBook > Product Catalog > Organic Chemistry > Carboxylic acids and derivatives > Target Protein-binding moiety 4
Target Protein-binding moiety 4
Target Protein-binding moiety 4 Basic information
- Product Name:
- Target Protein-binding moiety 4
- Synonyms:
-
- Target Protein-binding moiety 4
- PROTAC BRD4-binding moiety 2
- I-BET762 carboxylic acid
- GSK525762A carboxylic acid
- Molibresib carboxylic acid
- 4H-[1,2,4]Triazolo[4,3-a][1,4]benzodiazepine-4-acetic acid, 6-(4-chlorophenyl)-8-methoxy-1-methyl-, (4S)-
- I BET762 carboxylic acid,I-BET-762 carboxylic acid,IBET762 carboxylic acid
- (S)-2-(6-(4-Chlorophenyl)-8-methoxy-1-methyl-4H-benzo[f][1,2,4]triazolo[4,3-a][1,4]diazepin-4-yl)acetic acid
- CAS:
- 1300019-38-8
- MF:
- C20H17ClN4O3
- MW:
- 396.83
- Mol File:
- 1300019-38-8.mol
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Target Protein-binding moiety 4 Chemical Properties
- Boiling point:
- 648.3±65.0 °C(Predicted)
- Density
- 1.44±0.1 g/cm3(Predicted)
- storage temp.
- Store at -20°C
- solubility
- DMSO : 7.14 mg/mL (17.99 mM)
- form
- Solid
- pka
- 4.12±0.10(Predicted)
- color
- Light yellow to yellow
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Target Protein-binding moiety 4 Usage And Synthesis
Description
Target Protein-binding moiety 4 is a BRD4(1) inhibitor with an IC50 of 7.9 μM.
Target Protein-binding moiety 4 (compound 32) is a BRD4 (1) inhibitor with an IC50 of 7.9 μM[1].
References
[1]. Yifei Yang, et al. Combined pharmacophore models as virtual screening protocol against BRD4(1) inhibitor. Medicinal Chemistry Research (2016), 25(4), 585-595.
Target Protein-binding moiety 4Supplier
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