PD 135158 Chemical Properties

storage temp. 

Store at +4°C

solubility 

<61.68mg/ml in DMSO

PD 135158 Usage And Synthesis

Biological Activity

Potent and selective, nonpeptide CCK 2 receptor antagonist (IC 50 values are 2.8 and 1232 nM for CCK 2 and CCK 1 respectively) that displays negligible affinity at GABA A , benzodiazepine, substance P, neurotensin, opioid, bradykinin and 5-HT 3 receptors (IC 50 > 10 μ M). Exhibits anxiolytic activity in elevated plus maze and social interaction tests and increases food intake in rats.

PD 135158(130325-35-8)Related Product Information

• PD 135158
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