(2S)-2-AMINOPROPYL ESTER N2-[[2-(2-NAPHTHALENYL)-1H-BENZ[G]INDOL-3-YL]ACETYL]-D-LYSINE Chemical Properties

Boiling point:

827.9±65.0 °C(Predicted)

Density 

1.235±0.06 g/cm3(Predicted)

storage temp. 

Store at -20°C

solubility 

Soluble to 100 mM in DMSO

form 

Powder

pka

14.07±0.46(Predicted)

(2S)-2-AMINOPROPYL ESTER N2-[[2-(2-NAPHTHALENYL)-1H-BENZ[G]INDOL-3-YL]ACETYL]-D-LYSINE Usage And Synthesis

Uses

L-817,818 is a potent sst5 agonist.

Biological Activity

Potent and selective somatostatin sst 5 receptor agonist. K i values are 0.4, 3.3, 52, 64 and 82 nM for cloned human sst 5 , sst 1 , sst 2 , sst 3 and sst 4 receptors respectively. Inhibits growth hormone release from rat pituitary cells (EC 50 = 3.1 nM) and insulin release from mouse pancreatic islets (EC 50 = 0.3 nM) in vitro .

storage

Store at -20°C

(2S)-2-AMINOPROPYL ESTER N2-[[2-(2-NAPHTHALENYL)-1H-BENZ[G]INDOL-3-YL]ACETYL]-D-LYSINE(217480-27-8)Related Product Information

• 2-(2-NAPHTHYL)INDOLE
• INDOLE-3-ACETYL GLYCINE
• AC-D-LYS-OH
• (2S)-2-AMINOPROPYL ESTER N2-[[2-(2-NAPHTHALENYL)-1H-BENZ[G]INDOL-3-YL]ACETYL]-D-LYSINE