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ChemicalBook >  Product Catalog >  Pharmaceutical intermediates >  Bulk Drug Intermediates >  6-aMino-3-cyclopropyl-1-(2-fluoro-4-iodophenyl)pyriMidine-2,4(1H,3H)-dione

6-aMino-3-cyclopropyl-1-(2-fluoro-4-iodophenyl)pyriMidine-2,4(1H,3H)-dione

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6-aMino-3-cyclopropyl-1-(2-fluoro-4-iodophenyl)pyriMidine-2,4(1H,3H)-dione Basic information

Product Name:
6-aMino-3-cyclopropyl-1-(2-fluoro-4-iodophenyl)pyriMidine-2,4(1H,3H)-dione
Synonyms:
  • 6-Amino-3-cyclopropyl-1-(2-fluoro-4-iodophenyl)-1H-pyrimidine-2,4-dione
  • 6-amino-3-cyclopropyl-1-(2-fluoro-4-iodophenyl)pyrimidine-2,4-dione
  • 6-aMino-3-cyclopropyl-1-(2-fluoro-4-iodophenyl)pyriMidine-2,4(1H,3H)-dione
  • 2,4(1H,3H)-Pyrimidinedione, 6-amino-3-cyclopropyl-1-(2-fluoro-4-iodophenyl)-
  • 6-aMino-3-cyclopropyl-1-(2-fluoro-4-iodophenyl)pyriMidine-2,4(1H,3H)-dion
  • Trametinib Impurity 7
  • Olaquindox Impurity 7
  • Trametinib Impurity 02
CAS:
871700-28-6
MF:
C13H11FIN3O2
MW:
387.15
Mol File:
871700-28-6.mol
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6-aMino-3-cyclopropyl-1-(2-fluoro-4-iodophenyl)pyriMidine-2,4(1H,3H)-dione Chemical Properties

Boiling point:
449.1±55.0 °C(Predicted)
Density 
1.957±0.06 g/cm3(Predicted)
storage temp. 
2-8°C
pka
4.09±0.70(Predicted)
Appearance
Light yellow to yellow Solid
InChI
InChI=1S/C13H11FIN3O2/c14-9-5-7(15)1-4-10(9)18-11(16)6-12(19)17(13(18)20)8-2-3-8/h1,4-6,8H,2-3,16H2
InChIKey
WVVWGHZIHSJFNG-UHFFFAOYSA-N
SMILES
C1(=O)N(C2=CC=C(I)C=C2F)C(N)=CC(=O)N1C1CC1
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6-aMino-3-cyclopropyl-1-(2-fluoro-4-iodophenyl)pyriMidine-2,4(1H,3H)-dione Usage And Synthesis

Uses

6-Amino-3-cyclopropyl-1-(2-fluoro-4-iodophenyl)pyrimidine-2,4(1H,3H)-dione is a reagent used in the preparation of phenylpyrrolidines via C-H functionalization of amines with aryl halides by nickel-photoredox catalysis.

6-aMino-3-cyclopropyl-1-(2-fluoro-4-iodophenyl)pyriMidine-2,4(1H,3H)-dioneSupplier

Guangzhou Anyanren Pharmaceutical Technology Co., Ltd. Gold
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Daicel Chiral Technologies (China)CO.,LTD
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Tianjin Branch Chong pharmaceutical intermediates Co., Ltd.
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Shenzhen HwaGen Pharmaceutical Co.,Ltd
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