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Acalabrutinib Intermediate

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Acalabrutinib Intermediate Basic information

Product Name:
Acalabrutinib Intermediate
Synonyms:
  • Acalabrutinib Intermediate
  • acarabrutinib intermediate
  • (S)-4-(8-Amino-3-pyrrolidin-2-yl-imidazo[1,5-a]pyrazin-1-yl)-N- pyridin-2-yl-benzamide
  • Benzamide, 4-[8-amino-3-(2S)-2-pyrrolidinylimidazo[1,5-a]pyrazin-1-yl]-N-2-pyridinyl-
  • 4-[8-amino-3-(2S)-2-pyrrolidinylimidazo[1,5-a]pyrazin-1-yl]-N-2-pyridinyl-Benzamide
  • ACALABRUTINIB N-1
  • (S)-4-(8-Amino-3-pyrrolidin-2-yl-imidazo[1,5-a]pyrazin-1-yl)...
  • (S)-4-(8-amino-3-(pyrrolidin-2-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(pyridin-2-yl)benzamideQ: What is (S)-4-(8-amino-3-(pyrrolidin-2-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(pyridin-2-yl)benzamide Q: What is the CAS Number of (S)-4-(8-amino-3-(pyrrolidin-2-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(pyridin-2-yl)benzamide
CAS:
1420478-90-5
MF:
C22H21N7O
MW:
399.45
Product Categories:
  • Intermediates
Mol File:
1420478-90-5.mol
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Acalabrutinib Intermediate Chemical Properties

Density 
1.46±0.1 g/cm3(Predicted)
solubility 
DMSO (Slightly), Methanol (Slightly, Heated, Sonicated)
pka
11.47±0.70(Predicted)
form 
Solid
color 
Pale Beige to Beige
InChIKey
RWBYECCAYSUTDK-INIZCTEOSA-N
SMILES
C(NC1=NC=CC=C1)(=O)C1=CC=C(C2=C3N(C([C@@H]4CCCN4)=N2)C=CN=C3N)C=C1
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Acalabrutinib Intermediate Usage And Synthesis

Uses

4-[8-Amino-3-(2S)-2-pyrrolidinylimidazo[1,5-a]pyrazin-1-yl]-N-2-pyridinylbenzamide is a useful reagent for the preparation of nitrogen-containing heterocycle btk inhibitors.

Acalabrutinib IntermediateSupplier

Aurisco Pharmaceutical (Tianjin) Inc. Gold
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022-59885855
Sichuan Kaike Pharmaceutical Technology Co., Ltd Gold
Tel
13981731671
Email
checo@checopharma.com
ChengDu TongChuangYuan Pharmaceutical Co.Ltd
Tel
28-83379370 13880556291
Email
tcy@tcypharm.com
Nanjing Chemlin Chemical Co., Ltd
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025-83697070 13913916777;
Email
info@chemlin.com.cn
Daicel Chiral Technologies (China)CO.,LTD
Tel
021-50460086-9 15921403865
Email
han_yajun@dctc.daicel.com
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