N-type calcium channel blocker-1 Chemical Properties

Boiling point:

569.9±50.0 °C(Predicted)

Density 

1.013±0.06 g/cm3(Predicted)

storage temp. 

Store at -20°C

solubility 

Soluble in DMSO

pka

8.89±0.10(Predicted)

N-type calcium channel blocker-1 Usage And Synthesis

Uses

1-[[4-(Dimethylamino)phenyl]methyl]-N-[4-(3,3-dimethylbutyl)phenyl]-N-(3-methyl-2-buten-1-yl)-4-piperidinamine, is an N-type calcium channel blocker, and an orally active analgesic agent which shows high affinity to functionally block N-type calcium channels with an IC50 of 0.7 μM in the IMR32 assay.