Elismetrep
Elismetrep Basic information
- Product Name:
- Elismetrep
- Synonyms:
-
- Elismetrep
- Benzoic acid, 4-[[(4-cyclopropyl-3-isoquinolinyl)[[4-(trifluoromethoxy)phenyl]methyl]amino]sulfonyl]-
- CAS:
- 1400699-64-0
- MF:
- C27H21F3N2O5S
- MW:
- 542.53
- Mol File:
- 1400699-64-0.mol
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Elismetrep Chemical Properties
- form
- Solid
- color
- Off-white to light yellow
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Elismetrep Usage And Synthesis
Uses
Elismetrep (MT-8554) is an oral active TRPM8 inhibitor, and can be used for study of analgesic[1][2].
References
[1] Conklin M, et al. Neurokinin receptor antagonists as potential non-hormonal treatments for vasomotor symptoms of menopause. Ther Adv Reprod Health. 2023 Jun 22;17:26334941231177611. DOI:10.1177/26334941231177611
[2] Weyer AD, et al. Development of TRPM8 Antagonists to Treat Chronic Pain and Migraine. Pharmaceuticals (Basel). 2017 Mar 30;10(2):37. DOI:10.3390/ph10020037