PD 134308
PD 134308 Basic information
- Product Name:
- PD 134308
- Synonyms:
-
- PD 134308
- CI-988
- CAS:
- 130404-91-0
- MF:
- C42H59N5O11
- MW:
- 809.94476
- Mol File:
- 130404-91-0.mol
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PD 134308 Usage And Synthesis
Uses
CI-988 is a potent and selective cholecystokinin 2 (CCK-2) receptor antagonist that displays ~ 1600-fold selectivity over CCK1 receptors and has negligible affinity at other binding sites. CI-988 exhibits anxiolytic activity following oral administration. CI-98 inhibited the proliferation of small cell lung cancer (SCLC) cells in mice.