3-(1-METHYLPIPERIDIN-4-YL)-1H-INDOL-5-OL MALEATE
3-(1-METHYLPIPERIDIN-4-YL)-1H-INDOL-5-OL MALEATE Basic information
- Product Name:
- 3-(1-METHYLPIPERIDIN-4-YL)-1H-INDOL-5-OL MALEATE
- Synonyms:
-
- BRL 54443 MALEATE
- 3-(1-METHYLPIPERIDIN-4-YL)-1H-INDOL-5-OL MALEATE
- 3-(1-Methylpiperidin-4-yl)-1H-indol-5-ol maleate salt
- BRL 54443 maleate salt
- 1H-Indol-5-ol, 3-(1-methyl-4-piperidinyl)-, (2Z)-2-butenedioate (1:1)
- CAS:
- 1197333-54-2
- MF:
- C18H22N2O5
- MW:
- 346.38
- Product Categories:
-
- Serotonin receptor
- Mol File:
- Mol File
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3-(1-METHYLPIPERIDIN-4-YL)-1H-INDOL-5-OL MALEATE Chemical Properties
- storage temp.
- 2-8°C
- solubility
- H2O: 50 mg/mL
- form
- solid
- color
- white
- Water Solubility
- H2O: 50mg/mL
- InChI
- 1S/C14H18N2O.C4H4O4/c1-16-6-4-10(5-7-16)13-9-15-14-3-2-11(17)8-12(13)14;5-3(6)1-2-4(7)8/h2-3,8-10,15,17H,4-7H2,1H3;1-2H,(H,5,6)(H,7,8)/b;2-1-
- InChIKey
- INGCLXPSKXSYND-BTJKTKAUSA-N
- SMILES
- OC(=O)\C=C/C(O)=O.CN1CCC(CC1)c2c[nH]c3ccc(O)cc23
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MSDS
- Language:English Provider:SigmaAldrich
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3-(1-METHYLPIPERIDIN-4-YL)-1H-INDOL-5-OL MALEATE Usage And Synthesis
Uses
BRL 54443 Maleate Salt can be used in pharmacological activity and biological study of forskolin-free cAMP assay for Gi-coupled receptors.
Biological Activity
Potent 5-HT1E/1F serotonin receptor agonist.
in vivo
Reduction of flinching was considered as antinociception. Ipsilateral, but not contralateral, peripheral administration of BRL54443 (5-HT(1E/1F); 3-300 microg/paw) significantly reduced formalin-induced flinching in rats[3].
3-(1-METHYLPIPERIDIN-4-YL)-1H-INDOL-5-OL MALEATESupplier
Energy Chemical
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