Basic information Safety Supplier Related

N2-iso-Butyroyl-5'-(4,4'-dimethoxytrityl)-2'-O-propargylguanosine

Basic information Safety Supplier Related

N2-iso-Butyroyl-5'-(4,4'-dimethoxytrityl)-2'-O-propargylguanosine Basic information

Product Name:
N2-iso-Butyroyl-5'-(4,4'-dimethoxytrityl)-2'-O-propargylguanosine
Synonyms:
  • N2-iso-Butyroyl-5'-(4,4'-dimethoxytrityl)-2'-O-propargylguanosine
  • 5’-O-DMT-N2-isobutyryl-2’-O-propargylguanosine
  • N2-iso-Butyroyl-5’-O-(4,4’-dimethoxytrityl)-2’-O-propargylguanosine
  • Guanosine, 5'-O-[bis(4-methoxyphenyl)phenylmethyl]-N-(2-methyl-1-oxopropyl)-2'-O-2-propyn-1-yl-
  • 5'-O-DMT-2'-O-propargyl-N2-isobutyryl-guanosine
  • 5'-O-DMT-N2-isobutyryl-2'-O-propargylguanosine
CAS:
171486-53-6
MF:
C38H39N5O8
MW:
693.74496
Mol File:
171486-53-6.mol
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N2-iso-Butyroyl-5'-(4,4'-dimethoxytrityl)-2'-O-propargylguanosine Chemical Properties

Density 
1.31±0.1 g/cm3(Predicted)
pka
9.16±0.20(Predicted)
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N2-iso-Butyroyl-5'-(4,4'-dimethoxytrityl)-2'-O-propargylguanosine Usage And Synthesis

Uses

5'-O-DMT-N2-isobutyryl-2'-O-propargylguanosine is a guanosine analog. Some guanosine analogs have immunostimulatory activity. In some animal models, they also induce type I interferons, producing antiviral effects. Studies have shown that the functional activity of guanosine analogs is dependent on the activation of Toll-like receptor 7 (TLR7)[1].

References

[1] Lee J, et al. Molecular basis for the immunostimulatory activity of guanine nucleoside analogs: activation of Toll-like receptor 7. Proc Natl Acad Sci U S A. 2003 May 27;100(11):6646-51. DOI:10.1073/pnas.0631696100

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N2-iso-Butyroyl-5'-(4,4'-dimethoxytrityl)-2'-O-propargylguanosine(171486-53-6)Related Product Information