Pentanoic acid, 5-[(3-methoxypropyl)pentylamino]-4-[(2-naphthalenylsulfonyl)methyl]-5-oxo- Chemical Properties

Boiling point:

705.1±60.0 °C(Predicted)

Density 

1.187±0.06 g/cm3(Predicted)

storage temp. 

Store at -20°C

solubility 

Soluble in DMSO

pka

4.47±0.10(Predicted)

Pentanoic acid, 5-[(3-methoxypropyl)pentylamino]-4-[(2-naphthalenylsulfonyl)methyl]-5-oxo- Usage And Synthesis

Uses

CCK-A receptor inhibitor 1 is a cholecystokinin A (CCK-A) receptor inhibitor with a binging IC50 of 340 nM.

References

[1] Ajisawa Y, et al. [Studies on the synthesis of cholecystokinin A receptor antagonists. III. Synthesis and cholecystokinin A receptor inhibitory activities of naphthyl sulfone derivatives]. Yakugaku Zasshi. 1996 Aug;116(8):647-56. DOI:10.1248/yakushi1947.116.8_647