Basic information Safety Supplier Related

PD 168 077 MALEATE

Basic information Safety Supplier Related

PD 168 077 MALEATE Basic information

Product Name:
PD 168 077 MALEATE
Synonyms:
  • n-[[4-(2-cyanophenyl)-1-piperazinyl]methyl]-3-methylbenzamide maleate salt
  • pd 168,077 maleate salt
  • N-[[4-(2-Cyanophenyl)-1-piperazinyl]methyl]-3-methyl-benzamide
  • N-((4-(2-CYANOPHENYL)PIPERAZIN-1-YL)METHYL)-3-METHYLBENZAMIDE MALEATE
  • N-[[4-(2-cyanophenyl)piperazin-1-yl]methyl]-3-methylbenzamide
  • Benzamide, N-[[4-(2-cyanophenyl)-1-piperazinyl]methyl]-3-methyl-
  • 077
  • PD 168
CAS:
190383-31-4
MF:
C20H22N4O
MW:
334.41
Product Categories:
  • Dopamine receptor
Mol File:
190383-31-4.mol
More
Less

PD 168 077 MALEATE Chemical Properties

Boiling point:
554.6±50.0 °C(Predicted)
Density 
1.22±0.1 g/cm3(Predicted)
solubility 
DMSO: >10 mg/mL
form 
powder
pka
14.89±0.46(Predicted)
color 
white
InChIKey
NAEUGRPISCANHO-BTJKTKAUSA-N
SMILES
[H]\C(=C(/[H])C(O)=O)C(O)=O.Cc1cccc(c1)C(=O)NCN2CCN(CC2)c3ccccc3C#N
More
Less

Safety Information

Safety Statements 
22-24/25
WGK Germany 
3
Storage Class
11 - Combustible Solids
More
Less

PD 168 077 MALEATE Usage And Synthesis

Uses

The dopamine receptors play important role in cognition, memory, learning, and motor control (1). These receptors have been implicated as a therapeutic target for many psychiatric and neurological disorders. PD 168077 is a D4 dopamine receptor agonist and can be used to study ligand-receptor interactions of dopamine receptors (2).

Biological Activity

Selective D4 dopamine receptor agonist.

in vivo

PD-168077 (0.2-25.0 mg/kg) dose-dependently induces locomotion, which takes an unusual and characteristic ”shuffling” form with uncoordinated movements together with yawning, and episodes of myoclonic jerking; grooming, and rearing are reduced[1].

PD 168 077 MALEATESupplier

Chengdu YouSuo Biotechnology Limited
Tel
13693449011
Email
83948782@qq.com
Sigma-Aldrich
Tel
021-61415566 800-8193336
Email
orderCN@merckgroup.com
Tianjin Kailiqi Biotechnology Co., Ltd.
Tel
15076683720
Email
klq@cw-bio.com
Amadis Chemical Company Limited
Tel
571-89925085
Email
sales@amadischem.com
Nanjing KaiMubo Pharmaceutical Co., Ltd.
Tel
025-66162170
More
Less

PD 168 077 MALEATE(190383-31-4)Related Product Information