NALOXONE BENZOYLHYDRAZONE
NALOXONE BENZOYLHYDRAZONE Basic information
- Product Name:
- NALOXONE BENZOYLHYDRAZONE
- Synonyms:
-
- NALOXONE BENZOLYHYDRAZONE K3 OPIOID RECE PTOR AG
- [(5α)-4,5-epoxy-3,14-dihydroxy-17-(2-propenyl)morphinan-6-ylidene]hydrazide benzoic acid
- [(5alpha)-4,5-Epoxy-3,14-dihydroxy-17-(2-propenyl)morphinan-6-yliden]benzoic acid hydrazide
- [(5α)-4,5-Epoxy-3,14-dihydroxy-17-(2-propenyl)morphinan-6-ylidene]benzoicacidhydrazide
- NalBzoH
- Benzoic acid, 2-[(5α)-4,5-epoxy-3,14-dihydroxy-17-(2-propenyl)morphinan-6-ylidene]hydrazide
- Adamantane Impurity 48
- Benzoic acid, 2-[(5α)-4,5-epoxy-3,14-dihydroxy-17-(2-propenyl)morphinan-6-ylidene]hydrazide
- CAS:
- 119630-94-3
- MF:
- C26H27N3O4
- MW:
- 445.51
- Product Categories:
-
- Opioid receptor and opioid-like receptor
- Mol File:
- 119630-94-3.mol
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NALOXONE BENZOYLHYDRAZONE Chemical Properties
- Density
- 1.44±0.1 g/cm3(Predicted)
- storage temp.
- −20°C
- solubility
- DMSO: soluble
- form
- solid
- pka
- 9.11±0.40(Predicted)
- color
- yellow
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NALOXONE BENZOYLHYDRAZONE Usage And Synthesis
Biological Activity
Mixed opioid receptor agonist/antagonist. Acts as a potent and full agonist at κ , and a partial agonist at μ and δ opioid receptors (pEC 50 values are 9.45, 8.74 and 8.61 in a cAMP assay, 9.70, 8.59 and 8.49 in a [ 35 S]GTP γ S binding assay respectively). Fails to exert agonist effects at NOP receptors and antagonizes agonist-induced NOP activation. Stimulates κ -, μ - and δ -mediated analgesia and blocks NOP-induced supraspinal nociception.
NALOXONE BENZOYLHYDRAZONESupplier
3B Pharmachem (Wuhan) International Co.,Ltd.
- Tel
- 821-50328103-801 18930552037
- 3bsc@sina.com
EMMX Biotechnology LLC
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- 888-539-0666
- info@emmx.com
Shanghai EFE Biological Technology Co., Ltd.
- Tel
- 021-65675885 18964387627
- info@efebio.com
TargetMol Chemicals Inc.
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- +1-781-999-5354 +1-00000000000
- marketing@targetmol.com
cjbscvictory
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- 13348960310 13348960310
- 3003867561@qq.com