BQ-788
BQ-788 Basic information
- Product Name:
- BQ-788
- Synonyms:
-
- BQ-788 SODIUM
- BQ-788 SYNTHETIC >97% ETB ENDOTHELIN REC EPT
- N-[(cis-2,6-Dimethyl-1-piperidinyl)carbonyl]-4-methyl-L-leucyl-1-(methoxycarbonyl)-D-tryptophyl-D-norleucinesodiumsalt
- 1-ELAIDYLPHOSPHOCHOLINE, >97%
- N-[N-[N-[(2,6-Dimethyl-1-piperidinyl)carbonyl]-4-methyl-L-leucyl]-1-(methoxycarbonyl)-D-tryptophyl]-D-norleucine sodium salt, 2,6-Dimethylpiperidinecarbonyl-γ-Methyl-Leu-Nin-(Methoxycarbonyl)-D-Trp-D-Nle
- N-[N-[N-[(2,6-Dimethyl-1-piperidinyl)carbonyl]-
- DMpc-gaMMa-MeLeu-D-Trp(1-CO2CH3)-D-Nle.Na (DMpc : cis-2,6-DiMethylpiperidinocarbonyl)
- 2,6-Dimethylpiperidinecarbonyl-γ-Methyl-Leu-Nin-(Methoxycarbonyl)-D-Trp-D-Nle
- CAS:
- 156161-89-6
- MF:
- C34H52N5NaO7
- MW:
- 665.81
- Product Categories:
-
- Endothelin receptor
- Mol File:
- 156161-89-6.mol
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BQ-788 Chemical Properties
- storage temp.
- -20°C
- solubility
- acetonitrile: 0.3 mg/mL
- form
- solid
- color
- white
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BQ-788 Usage And Synthesis
Uses
BQ-788 has been used as a selective endothelin-B (ETRB) blocker in human airway smooth muscle cells (HASMCs), uterine mesothelial cells (UtMCs)-derived vascular smooth muscle cells (VSMCs), and human umbilical vein endothelial cells (HUVECs)
Biological Activity
Potent, selective ET B receptor antagonist (IC 50 = 1.2 nM for inhibition of ET-1 binding to human Girardi heart cells).
Biochem/physiol Actions
Selective ETB endothelin receptor antagonist.
storage
+4°C
BQ-788Supplier
Hangzhou Sinoda Pharmaceutical Technology Co. LTD Gold
- Tel
- 17306812703
- 3007955328@qq.com
3B Pharmachem (Wuhan) International Co.,Ltd.
- Tel
- 821-50328103-801 18930552037
- 3bsc@sina.com
Shanghai Sinch Parmaceuticals Tech. Co. Ltd.
- Tel
- +86-21-54098501
- sales@sinch.com.cn
Chemsky（shanghai）International Co.,Ltd.
- Tel
- 021-50135380
- shchemsky@sina.com
Haoyuan Chemexpress Co., Ltd.
- Tel
- 021-58950125
- info@chemexpress.com