Milameline Chemical Properties

Boiling point:

221.1±50.0 °C(Predicted)

Density 

1.00±0.1 g/cm3(Predicted)

storage temp. 

Desiccate at -20°C

pka

8.22±0.40(Predicted)

Milameline Usage And Synthesis

Uses

Antidementia (partial muscarinic agonist.

Uses

Milameline is a muscarinic receptor agonist.

Biological Activity

Muscarinic receptor agonist that displays roughly equal affinity at all receptor subtypes (K i values are 2.3, 2.4, 3.6, 3.8 and 4.3 μ M for hM 1 , hM 2 , hM 3 , hM 4 and hM 5 receptors respectively). Cognitive enhancer; reverses spatial memory deficits in rats.

Milameline(139886-32-1)Related Product Information

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• Milameline
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