RX 809055AX
RX 809055AX Basic information
- Product Name:
- RX 809055AX
- Synonyms:
-
- RX 809055AX
- CAS:
- 122566-12-5
- MF:
- C29H29ClN2O4
- MW:
- 505.00456
- Mol File:
- 122566-12-5.mol
More
Less
RX 809055AX Usage And Synthesis
Description
RX 809055AX is a long lasting opioid antagonist at mu and delta receptors.
Uses
RX 809055AX is a potent long lasting opioid antagonist with selectivity towards at mu and delta receptors[1].
IC 50
μ Opioid Receptor/MOR; δ Opioid Receptor/DOR
References
[1] Lemcke PK, Ayres EA, Kramer TH, Burks TF. RX809055AX in vivo: a long lasting opioid antagonist at mu and delta receptors. Proc West Pharmacol Soc. 1989;32:173-5. PMID:2550942