CaproMorelin Tartrate

Product Name: CaproMorelin Tartrate
CAS No.: 193273-69-7
Chemical Name: CaproMorelin Tartrate
Synonyms: CS-2136;CP 424391-18;CP-424391 tartrate;CaproMorelin Tartrate;CP 424391-18; CP-424391 TARTRATE;Capromorelin tartrate (CP-424,391);Capromorelin Tartrate, 10 mM in DMSO;Inhibitor,Growth hormone secretagogue receptor,GHSR,Capromorelin,inhibit,Capromorelin Tartrate;N-{2-[(3aS)-3a-benzyl-2-methyl-3-methylidene-2,3,3a,4,6,7-hexahydro-5H-pyrazolo[4,3-c]pyridin-5-yl]-1-(benzyloxy)-2-oxoethyl}-2-methylalaninamide 2,3-dihydroxybutanedioate (1:1);2-amino-N-((R)-1-((R)-3a-benzyl-2-methyl-3-oxo-3a,4,6,7-tetrahydro-2H-pyrazolo[4,3-c]pyridin-5(3H)-yl)-3-(benzyloxy)-1-oxopropan-2-yl)-2-methylpropanamide (2R,3R)-2,3-dihydroxysuccinate
CBNumber: CB02611352
Molecular Formula: C32H41N5O10
Formula Weight: 655.71
MOL File: 193273-69-7.mol

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CaproMorelin Tartrate Property

Melting point:: >150oC (dec.)
storage temp.: Hygroscopic, -20°C Freezer, Under inert atmosphere
solubility: DMSO (Slightly), Methanol (Slightly)
form: Solid
color: White to Light Yellow
Water Solubility: H2O: 20mg/mL, clear
Stability:: Hygroscopic

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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word: Warning

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N-Bromosuccinimide Price

TRC

Product number: C175645
Product name: CapromorelinTartrate
Packaging: 1mg
Price: $50
Updated: 2021/12/16

TRC

Product number: C175645
Product name: CapromorelinTartrate
Packaging: 25mg
Price: $265
Updated: 2021/12/16

TRC

Product number: C175645
Product name: CapromorelinTartrate
Packaging: 100mg
Price: $780
Updated: 2021/12/16

ChemScene

Product number: CS-6929
Product name: CapromorelinTartrate
Purity: 98.19%
Packaging: 2mg
Price: $50
Updated: 2021/12/16

ChemScene

Product number: CS-6929
Product name: CapromorelinTartrate
Purity: 98.19%
Packaging: 50mg
Price: $460
Updated: 2021/12/16

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CaproMorelin Tartrate Chemical Properties,Usage,Production

Uses

Treatment and prevention of frailty; treatment of congestive heart failure; treatment of catabolic illness (growth hormone secretagogue).

Uses

Capromorelin Tartrate acts as a reagent used in the preparation of pyrazolopyridine amide growth hormone secretagogues for treatment of fibromyalgia

Biological Activity

Capromorelin tartrate is a potent ghrelin receptor agonist/growth hormone secretagogue (Ki = 7 nM). In r at pituitary cells, Capromorlelin incudes growth hormone (GH) secretion with an EC50 of 3 nM. Capromorelin also increases gastric motility and has been studied recently in patients with spinal cord injuries.

in vivo

Dogs receiving capromorelin (30 mg/mL) have food consumption that is significantly greater than dogs treated with placebo. All dogs in the capromorelin group gain weight by 0.52 kg, more than that of placebo group^[1]. Capromorelin shows enhanced intestinal absorption in rodent models and exhibits superior pharmacokinetic properties, including high bioavailabilities in two animal species [F(rat)=65%, F(dog)=44%]^[2]. Capromorelin stimulates GH release in anesthesized rat model, with ED₅₀ of 0.05 mg/kg iv^[2].

CaproMorelin Tartrate Preparation Products And Raw materials

Raw materials

Preparation Products

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CaproMorelin Tartrate Suppliers

China 73 India 1 United States 9 Global 83

BEIJING QIONGFENG TECHNOLOGICAL CO., LTD.

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Shijiazhuang Molechem PharmaTech Co.Ltd

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MedChemexpress LLC

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193273-69-7, CaproMorelin TartrateRelated Search:

CaproMorelin Tartrate

CP 424391-18

CP 424391-18; CP-424391 TARTRATE

CP-424391 tartrate

CS-2136

N-{2-[(3aS)-3a-benzyl-2-methyl-3-methylidene-2,3,3a,4,6,7-hexahydro-5H-pyrazolo[4,3-c]pyridin-5-yl]-1-(benzyloxy)-2-oxoethyl}-2-methylalaninamide 2,3-dihydroxybutanedioate (1:1)

Capromorelin tartrate (CP-424,391)

Inhibitor,Growth hormone secretagogue receptor,GHSR,Capromorelin,inhibit,Capromorelin Tartrate

2-amino-N-((R)-1-((R)-3a-benzyl-2-methyl-3-oxo-3a,4,6,7-tetrahydro-2H-pyrazolo[4,3-c]pyridin-5(3H)-yl)-3-(benzyloxy)-1-oxopropan-2-yl)-2-methylpropanamide (2R,3R)-2,3-dihydroxysuccinate

Capromorelin Tartrate, 10 mM in DMSO

193273-69-7

C28H35N5O4C4H6O6

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