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5-BroMo-3-Methylpyrazin-2-ol

Product Name
5-BroMo-3-Methylpyrazin-2-ol
CAS No.
100047-56-1
Chemical Name
5-BroMo-3-Methylpyrazin-2-ol
Synonyms
5-BroMo-3-Methylpyrazin-2-ol;5-BroMo-3-Methylpyrazin-2-one;5-bromo-3-methyl-1H-pyrazin-2-one;5-Bromo-3-methyl-2(1H)-pyrazinone;2(1H)-Pyrazinone, 5-bromo-3-methyl;5-BroMo-2-hydroxy-3-Methyl pyrazine
CBNumber
CB02661100
Molecular Formula
C5H5BrN2O
Formula Weight
189.01
MOL File
100047-56-1.mol
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5-BroMo-3-Methylpyrazin-2-ol Property

Density 
1.84±0.1 g/cm3(Predicted)
storage temp. 
under inert gas (nitrogen or Argon) at 2-8°C
pka
10.05±0.60(Predicted)
Appearance
Light yellow to yellow Solid
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Warning
Hazard statements

H302Harmful if swallowed

H315Causes skin irritation

H319Causes serious eye irritation

H332Harmful if inhaled

H335May cause respiratory irritation

Precautionary statements

P280Wear protective gloves/protective clothing/eye protection/face protection.

P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

P310Immediately call a POISON CENTER or doctor/physician.

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N-Bromosuccinimide Price

Biosynth Carbosynth
Product number
FB145035
Product name
5-Bromo-2-hydroxy-3-methyl pyrazine
Packaging
25mg
Price
$100
Updated
2021/12/16
Biosynth Carbosynth
Product number
FB145035
Product name
5-Bromo-2-hydroxy-3-methyl pyrazine
Packaging
50mg
Price
$150
Updated
2021/12/16
AK Scientific
Product number
1452CZ
Product name
5-Bromo-3-methylpyrazin-2-ol
Packaging
1g
Price
$188
Updated
2021/12/16
Biosynth Carbosynth
Product number
FB145035
Product name
5-Bromo-2-hydroxy-3-methyl pyrazine
Packaging
100mg
Price
$200
Updated
2021/12/16
Biosynth Carbosynth
Product number
FB145035
Product name
5-Bromo-2-hydroxy-3-methyl pyrazine
Packaging
250mg
Price
$300
Updated
2021/12/16
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5-BroMo-3-Methylpyrazin-2-ol Chemical Properties,Usage,Production

Synthesis

19838-07-4

100047-56-1

The general procedure for the synthesis of 2-hydroxy-3-methyl-5-bromopyrazine from 2-hydroxy-3-methylpyrazine was as follows: to a solution of 3-methylpyrazin-2-ol (1.5 g, 13.62 mmol) in anhydrous N,N-dimethylformamide (DMF, 20 mL) was added batchwise at 0 °C N-bromosuccinimide (NBS, 2.67 g, 14.98 mmol). The reaction mixture was slowly warmed to room temperature and stirred overnight. Upon completion of the reaction, the mixture was poured into ice water and extracted with a solvent mixture of isopropanol (IPA)/dichloromethane (DCM, 1/5, v/v). The organic phases were combined, dried with anhydrous sodium sulfate (Na2SO4), filtered and concentrated under reduced pressure. The crude product was purified by silica gel column chromatography with 80% ethyl acetate/hexane (v/v) as eluent to afford 2-hydroxy-3-methyl-5-bromopyrazine as white solid (1.97 g, 10.42 mmol, 77% yield). The product was analyzed by mass spectrometry (LCMS) with measured m/z = 189.0 [M+H]+ (calculated exact mass of C5H5BrN2O: 188.0).1H NMR (400 MHz, DMSO-d6) δppm: 2.27 (d, J = 0.5 Hz, 3H), 7.73 (s, 1H), 12.3 (s, 1H).

References

[1] Patent: WO2011/127051, 2011, A1. Location in patent: Page/Page column 205

5-BroMo-3-Methylpyrazin-2-ol Preparation Products And Raw materials

Raw materials

Preparation Products

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5-BroMo-3-Methylpyrazin-2-ol Suppliers

Shanghai Hanhong Scientific Co.,Ltd.
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100047-56-1, 5-BroMo-3-Methylpyrazin-2-olRelated Search:


  • 5-BroMo-3-Methylpyrazin-2-ol
  • 5-BroMo-3-Methylpyrazin-2-one
  • 5-BroMo-2-hydroxy-3-Methyl pyrazine
  • 2(1H)-Pyrazinone, 5-bromo-3-methyl
  • 5-Bromo-3-methyl-2(1H)-pyrazinone
  • 5-bromo-3-methyl-1H-pyrazin-2-one
  • 100047-56-1