ChemicalBook > CAS DataBase List > glucagon receptor antagonists-4
glucagon receptor antagonists-4
- Product Name
- glucagon receptor antagonists-4
- CAS No.
- 1393124-08-7
- Chemical Name
- glucagon receptor antagonists-4
- Synonyms
- CS-2641;PF6291874;GCGR-IN-17;PF-06291874 >=98% (HPLC);Glucagon Receptor Antagonist 4;lucagon receptor antagonists-4;glucagon receptor antagonists-4;PF06291874;PF-06291874;PF 06291874;PF-06291874(glucagon receptor antagonists-4);N-{4-[(1S)-1-{3,5-Dimethyl-4-[4-(trifluoromethyl)-1H-pyrazol-1-yl]phenoxy}butyl]benzoyl}-β-alanine
- CBNumber
- CB03133347
- Molecular Formula
- C26H28F3N3O4
- Formula Weight
- 503.51
- MOL File
- 1393124-08-7.mol
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glucagon receptor antagonists-4 Property
- Boiling point:
- 675.0±55.0 °C(Predicted)
- Density
- 1.27±0.1 g/cm3(Predicted)
- storage temp.
- Store at -20°C
- solubility
- DMF: 50mg/mL; DMSO: 50mg/mL; DMSO:PBS (pH 7.2) (1:1): 0.5mg/mL; Ethanol: 0.5mg/mL
- form
- A crystalline solid
- pka
- 4.28±0.10(Predicted)
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Safety
- HS Code
- 2933998090
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Hazard and Precautionary Statements (GHS)
- Symbol(GHS)
-
- Signal word
- Warning
- Hazard statements
-
H302Harmful if swallowed
H315Causes skin irritation
H319Causes serious eye irritation
H335May cause respiratory irritation
- Precautionary statements
-
P261Avoid breathing dust/fume/gas/mist/vapours/spray.
P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.
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N-Bromosuccinimide Price
Cayman Chemical
- Product number
- 22164
- Product name
- Glucagon Receptor Antagonist 4
- Packaging
- 1mg
- Price
- $32
- Updated
- 2024/03/01
Cayman Chemical
- Product number
- 22164
- Product name
- Glucagon Receptor Antagonist 4
- Packaging
- 5mg
- Price
- $93
- Updated
- 2024/03/01
Cayman Chemical
- Product number
- 22164
- Product name
- Glucagon Receptor Antagonist 4
- Packaging
- 10mg
- Price
- $169
- Updated
- 2024/03/01
Cayman Chemical
- Product number
- 22164
- Product name
- Glucagon Receptor Antagonist 4
- Packaging
- 25mg
- Price
- $381
- Updated
- 2024/03/01
TRC
- Product number
- P294103
- Product name
- PF-06291874
- Packaging
- 10mg
- Price
- $315
- Updated
- 2021/12/16
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glucagon receptor antagonists-4 Chemical Properties,Usage,Production
Uses
PF-06291874 is a novel and potent glucagon receptor antagonist for the potential treatment of diabetes mellitus. PF-06291874, has a lower molcular weight and lipophilicity than historical glucagon receptor antagonists, resulting in excellent selectivity in broad-panel screening, lower cytotoxicity, and excellent overall in vivo safety in early pre-clinical testing.
glucagon receptor antagonists-4 Preparation Products And Raw materials
Raw materials
Preparation Products
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