ChemicalBook > CAS DataBase List > CY 208-243

CY 208-243

Product Name
CY 208-243
CAS No.
100999-26-6
Chemical Name
CY 208-243
Synonyms
CY 208-243;CY 208243,CY 208 243;(6aR)-4,6,6aα,7,8,12bβ-Hexahydro-7-methylindolo[4,3-ab]phenanthridine;(6aα,12bβ)-4,6,6a,7,8,12b-Hexahydro-7-methylindolo[4,3-ab]phenanthridine;(6aR,12bβ)-4,6,6a,7,8,12b-Hexahydro-7-methylindolo[4,3-ab]phenanthridine;(-)-(6AR,12BR)-4,6,6A,7,8,12B-HEXAHYDRO-7-METHYLINDOLO[4,3-A]PHENANTHRIDIN;(-)-(6aR,12bR)-4,6,6a,7,8,12β-Hexahydro-7-methylindolo[4,3-a]phenanthridin;[6aR,12bR,(-)]-4,6,6a,7,8,12b-Hexahydro-7-methylindolo[4,3-ab]phenanthridine;Indolo[4,3-ab]phenanthridine, 4,6,6a,7,8,12b-hexahydro-7-methyl-, (6aR,12bR)-
CBNumber
CB0461748
Molecular Formula
C19H18N2
Formula Weight
274.36
MOL File
100999-26-6.mol
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CY 208-243 Property

Boiling point:
466.5±33.0 °C(Predicted)
Density 
1.225±0.06 g/cm3(Predicted)
storage temp. 
Store at RT
solubility 
Soluble to 100 mM in DMSO
form 
Powder
pka
17.40±0.20(Predicted)
color 
White to off-white
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Hazard and Precautionary Statements (GHS)

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N-Bromosuccinimide Price

Tocris
Product number
1249
Product name
CY208-243
Packaging
10
Price
$212
Updated
2021/12/16
Tocris
Product number
1249
Product name
CY208-243
Packaging
50
Price
$870
Updated
2021/12/16
TRC
Product number
C991923
Product name
CY208-243
Packaging
10mg
Price
$170
Updated
2021/12/16
TRC
Product number
C991923
Product name
CY208-243
Packaging
25mg
Price
$335
Updated
2021/12/16
ChemScene
Product number
CS-0024842
Product name
CY208-243
Purity
99.78%
Packaging
1mg
Price
$145
Updated
2021/12/16
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CY 208-243 Chemical Properties,Usage,Production

Uses

CY 208-243 is a selective D1DR receptor agonist.

Definition

ChEBI: LSM-3788 is a member of phenanthridines.

Biological Activity

Centrally active dopamine D 1 receptor agonist, selective over D 2 receptor sites. Stimulates adenylate cyclase in rat striatal homogenates with an EC 50 of 125 nM. Unlike SKF 38393 ((?-1-Phenyl-2,3,4,5-tetrahydro-(1H)-3-benzazepine-7,8-diol hydrobromide ), it exerts anti-Parkinsonian activity in animal models.

in vivo

Pretreatment with CY 208-243 (2.5 mg/kg; s.c.) prevents the increase of DA release and metabolism induced by the D-1 antagonist, SCH 23390 (0.05 mg/kg; s.c.)[1].

Animal Model:Male Sprague-Dawley rats (180-200 g)[1]
Dosage:2.5 mg/kg
Administration:Subcutaneous
Result:Prevented the increase of DA release and metabolism induced by the D-1 antagonist.

IC 50

D1 Receptor

storage

Store at RT

CY 208-243 Preparation Products And Raw materials

Raw materials

Preparation Products

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CY 208-243 Suppliers

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100999-26-6, CY 208-243Related Search:

Phenanthridine CY 208-243 [2-(1 H-INDOL-3-YL)-ETHYL]-(2-METHYL-BENZYL)-AMINE

  • (-)-(6AR,12BR)-4,6,6A,7,8,12B-HEXAHYDRO-7-METHYLINDOLO[4,3-A]PHENANTHRIDIN
  • (6aR)-4,6,6aα,7,8,12bβ-Hexahydro-7-methylindolo[4,3-ab]phenanthridine
  • (6aR,12bβ)-4,6,6a,7,8,12b-Hexahydro-7-methylindolo[4,3-ab]phenanthridine
  • (6aα,12bβ)-4,6,6a,7,8,12b-Hexahydro-7-methylindolo[4,3-ab]phenanthridine
  • [6aR,12bR,(-)]-4,6,6a,7,8,12b-Hexahydro-7-methylindolo[4,3-ab]phenanthridine
  • (-)-(6aR,12bR)-4,6,6a,7,8,12β-Hexahydro-7-methylindolo[4,3-a]phenanthridin
  • CY 208-243
  • Indolo[4,3-ab]phenanthridine, 4,6,6a,7,8,12b-hexahydro-7-methyl-, (6aR,12bR)-
  • CY 208243,CY 208 243
  • 100999-26-6
  • Dopamine receptor