ChemicalBook > CAS DataBase List > Protac linker 5
Protac linker 5
- Product Name
- Protac linker 5
- CAS No.
- 2245697-83-8
- Chemical Name
- Protac linker 5
- Synonyms
- Protac linker 5;(S,R,S)-AHPC-C3-NH2;VH032-C4-NH2 hydrochloride;VHL Ligand-Linker Conjugates 13;E3 ligase Ligand-Linker Conjugates 28;inhibit,E3 Ligase Ligand-Linker Conjugates,(S,R,S)AHPCC4NH2 hydrochloride,Inhibitor,(S,R,S) AHPC C4 NH2 hydrochloride
- CBNumber
- CB04845049
- Molecular Formula
- C27H40ClN5O4S
- Formula Weight
- 566.16
- MOL File
- 2245697-83-8.mol
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Protac linker 5 Property
- form
- Solid
- color
- Light yellow to green yellow
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Protac linker 5 Chemical Properties,Usage,Production
Uses
(S,R,S)-AHPC-C4-NH2 hydrochloride is a synthesized E3 ligase ligand-linker conjugate that incorporates the (S,R,S)-AHPC based VHL ligand and a linker used for EED-Targeted PROTAC[1].
IC 50
VHL
References
[1] Hsu JH, et al. EED-Targeted PROTACs Degrade EED, EZH2, and SUZ12 in the PRC2 Complex. Cell Chem Biol. 2019 Nov 26. pii: S2451-9456(19)30362-9. DOI:10.1016/j.chembiol.2019.11.004
Protac linker 5 Preparation Products And Raw materials
Raw materials
Preparation Products
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Protac linker 5 Suppliers
- Tel
- +1-781-999-5354; +17819995354
- marketing@targetmol.com
- Country
- United States
- ProdList
- 32435
- Advantage
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