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amauromine

Product Name
amauromine
CAS No.
88360-87-6
Chemical Name
amauromine
Synonyms
WF-6237;FR-900220;amauromine;Antibiotic FR-900220;4'',5'':1',5']dipyrrolo[2,3-b:2',3'-b']diindole-7,15(5H,7aH)-dione;4a-bromo-8-methoxy-1,4a,5,10a-tetrahydropyrimido[5,4-b]quinoline-2,4,10(3h)-trione;(5aS,7aS,8aR,13aS,15aS,16aR)-8a,16a-Bis(1,1-dimethyl-2-propen-1-yl)-5a,8,8a,13,13a,15a,16,16a-octahydro-pyrazino[1'',2'':1,5;(5aS)-8aα,16aα-Bis(1,1-dimethyl-2-propenyl)-5aα,8,8a,13,13aα,15aβ,16,16a-octahydropyrazino[1'',2'':1,5:4'',5'':1',5']dipyrrolo[2,3-b:2',3'-b']diindole-7,15(5H,7aβH)-dione;4'',5'':1',5']dipyrrolo[2,3-b:2',3'-b']diindole-7,15(5H,7aH)-dione, 8a,16a-bis(1,1-dimethyl-2-propen-1-yl)-5a,8,8a,13,13a,15a,16,16a-octahydro-, (5aS,7aS,8aR,13aS,15aS,16aR)-
CBNumber
CB11327574
Molecular Formula
C32H36N4O2
Formula Weight
508.662
MOL File
88360-87-6.mol
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amauromine Property

Boiling point:
689.9±55.0 °C(Predicted)
Density 
1.28±0.1 g/cm3(Predicted)
storage temp. 
Store at -20°C
solubility 
DMSO: Soluble; Ethanol: Soluble; Methanol: Soluble
form 
A solid
pka
3.26±0.60(Predicted)
color 
Brown
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Safety

Toxicity
LD50 intraperitoneal in mouse: > 200mg/kg
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Warning
Precautionary statements

P261Avoid breathing dust/fume/gas/mist/vapours/spray.

P264Wash hands thoroughly after handling.

P264Wash skin thouroughly after handling.

P270Do not eat, drink or smoke when using this product.

P271Use only outdoors or in a well-ventilated area.

P280Wear protective gloves/protective clothing/eye protection/face protection.

P301+P312IF SWALLOWED: call a POISON CENTER or doctor/physician IF you feel unwell.

P302+P352IF ON SKIN: wash with plenty of soap and water.

P304+P340IF INHALED: Remove victim to fresh air and Keep at rest in a position comfortable for breathing.

P321Specific treatment (see … on this label).

P330Rinse mouth.

P501Dispose of contents/container to..…

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N-Bromosuccinimide Price

Cayman Chemical
Product number
23886
Product name
Amauromine
Purity
≥98%
Packaging
250μg
Price
$79
Updated
2024/03/01
Cayman Chemical
Product number
23886
Product name
Amauromine
Purity
≥98%
Packaging
1mg
Price
$219
Updated
2024/03/01
Usbiological
Product number
044497
Product name
Amauromine
Packaging
250ug
Price
$290
Updated
2021/12/16
TRC
Product number
A575993
Product name
Amauromine
Packaging
2.5mg
Price
$295
Updated
2021/12/16
American Custom Chemicals Corporation
Product number
INB0003887
Product name
AMAUROMINE
Purity
95.00%
Packaging
5MG
Price
$501.22
Updated
2021/12/16
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amauromine Chemical Properties,Usage,Production

Description

Amauromine is a neutral antagonist of the cannabinoid (CB) receptor CB1 that is selective for CB1 (Ki = 178 nM; Kb = 66.6 nM) over CB2, with no activity at CB2 receptors at concentrations up to 10 μM. It is also an antagonist of GPR18 (IC50 = 3.74 μM). Amauromine has vasodilatory activity.

Uses

Amauromine is a CB1 and Calcium Channel antagonist.

storage

+4°C

amauromine Preparation Products And Raw materials

Raw materials

Preparation Products

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amauromine Suppliers

China 20 India 1 United Kingdom 1 United States 4 Global 26
TargetMol Chemicals Inc.
Tel
+1-781-999-5354 +1-00000000000
Email
marketing@targetmol.com
Country
United States
ProdList
32165
Advantage
58
Cayman Chemical Company
Tel
--
Fax
--
Email
cayman@caymanchem.com
Country
United States
ProdList
6213
Advantage
81
United States Biological
Tel
--
Fax
--
Email
chemicals@usbio.net
Country
United States
ProdList
6214
Advantage
80
Santa Cruz Biotechnology, Inc.
Tel
--
Fax
--
Email
scbt@scbt.com
Country
United States
ProdList
3597
Advantage
60

88360-87-6, amauromineRelated Search:

(R)-HEXAHYDROPYRROLO[1,2-A]PYRAZIN-1(2H)-ONE CYCLO(-LEU-GLY) 2-(3-PHENYL-PYRROLIDIN-1-YL)-ETHYLAMINE CHEMBRDG-BB 4012298 Piperazinone, 1-butyl- (9CI) CYCLO(-LEU-PRO) Pyrrolo[1,2-a]pyrazine, octahydro-3-isobutyl- (5CI) N-(1-METHYL-3-PHENYLPROPYL)-N-VALERAMIDE CYCLO(-GLY-PRO) amauromine 1H-Indol-2-amine 3-ISOBUTYL-6-METHYL-2,5-PIPERAZINEDIONE

  • amauromine
  • (5aS)-8aα,16aα-Bis(1,1-dimethyl-2-propenyl)-5aα,8,8a,13,13aα,15aβ,16,16a-octahydropyrazino[1'',2'':1,5:4'',5'':1',5']dipyrrolo[2,3-b:2',3'-b']diindole-7,15(5H,7aβH)-dione
  • Antibiotic FR-900220
  • FR-900220
  • WF-6237
  • (5aS,7aS,8aR,13aS,15aS,16aR)-8a,16a-Bis(1,1-dimethyl-2-propen-1-yl)-5a,8,8a,13,13a,15a,16,16a-octahydro-pyrazino[1'',2'':1,5
  • 4'',5'':1',5']dipyrrolo[2,3-b:2',3'-b']diindole-7,15(5H,7aH)-dione
  • 4'',5'':1',5']dipyrrolo[2,3-b:2',3'-b']diindole-7,15(5H,7aH)-dione, 8a,16a-bis(1,1-dimethyl-2-propen-1-yl)-5a,8,8a,13,13a,15a,16,16a-octahydro-, (5aS,7aS,8aR,13aS,15aS,16aR)-
  • 4a-bromo-8-methoxy-1,4a,5,10a-tetrahydropyrimido[5,4-b]quinoline-2,4,10(3h)-trione
  • 88360-87-6
  • C32H36N4O2