3-AMINO-N-[(4-CHLOROPHENYL)METHYL]-4,6-DIMETHYLTHIENO[2,3-B]PYRIDINE-2-CARBOXAMIDE
- Product Name
- 3-AMINO-N-[(4-CHLOROPHENYL)METHYL]-4,6-DIMETHYLTHIENO[2,3-B]PYRIDINE-2-CARBOXAMIDE
- CAS No.
- 633283-39-3
- Chemical Name
- 3-AMINO-N-[(4-CHLOROPHENYL)METHYL]-4,6-DIMETHYLTHIENO[2,3-B]PYRIDINE-2-CARBOXAMIDE
- Synonyms
- VU 10010;3-Amino-N-(4-chlorobenzyl)-4,6-dimethylthieno[2,3-b]pyridine-2-carboxamide;3-Amino-4,6-dimethyl-thieno[2,3-b]pyridine-2-carboxylic acid 4-chloro-benzylamide;3-AMINO-N-[(4-CHLOROPHENYL)METHYL]-4,6-DIMETHYLTHIENO[2,3-B]PYRIDINE-2-CARBOXAMIDE;Thieno[2,3-b]pyridine-2-carboxamide, 3-amino-N-[(4-chlorophenyl)methyl]-4,6-dimethyl-;hippocampus,synapses,acetylcholine,allosteric,excitatory,transmission,mAChR,Muscarinic acetylcholine receptor,carbachol,Inhibitor,inhibit,VU10010,proteins,depression,VU-10010
- CBNumber
- CB12448258
- Molecular Formula
- C17H16ClN3OS
- Formula Weight
- 345.85
- MOL File
- 633283-39-3.mol
3-AMINO-N-[(4-CHLOROPHENYL)METHYL]-4,6-DIMETHYLTHIENO[2,3-B]PYRIDINE-2-CARBOXAMIDE Property
- storage temp.
- Store at +4°C
- solubility
- Soluble in DMSO > 10 mM
- form
- Powder
- color
- White to off-white
Hazard and Precautionary Statements (GHS)
- Symbol(GHS)
-
- Signal word
- Danger
- Hazard statements
-
H301Toxic if swalloed
H319Causes serious eye irritation
- Precautionary statements
-
P264Wash hands thoroughly after handling.
P264Wash skin thouroughly after handling.
P270Do not eat, drink or smoke when using this product.
P280Wear protective gloves/protective clothing/eye protection/face protection.
P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.
P337+P313IF eye irritation persists: Get medical advice/attention.
P405Store locked up.
P501Dispose of contents/container to..…
N-Bromosuccinimide Price
- Product number
- 3141
- Product name
- VU10010
- Purity
- ≥99%(HPLC)
- Packaging
- 10
- Price
- $197
- Updated
- 2021/12/16
- Product number
- 3141
- Product name
- VU10010
- Purity
- ≥99%(HPLC)
- Packaging
- 50
- Price
- $780
- Updated
- 2021/12/16
- Product number
- 257070
- Product name
- VU 10010
- Packaging
- 10mg
- Price
- $446
- Updated
- 2021/12/16
- Product number
- A603825
- Product name
- 3-Amino-N-[(4-chlorophenyl)methyl]-4,6-dimethylthieno[2,3-b]pyridine-2-carboxamide
- Packaging
- 10mg
- Price
- $130
- Updated
- 2021/12/16
- Product number
- B7285
- Product name
- VU10010
- Packaging
- 10mg
- Price
- $297
- Updated
- 2021/12/16
3-AMINO-N-[(4-CHLOROPHENYL)METHYL]-4,6-DIMETHYLTHIENO[2,3-B]PYRIDINE-2-CARBOXAMIDE Chemical Properties,Usage,Production
Uses
This compound acts as a selective allosteric M4 (Muscarinic Acetylcholine Receptor) agonist.
Biological Activity
Selective allosteric potentiator of M 4 acetylcholine receptors (EC 50 values are 33 and 0.7 nM for ACh in the absence and presence of VU10010 espectively). Binds to an allosteric site on the receptor increasing affinity for ACh and coupling to G-proteins.
storage
Store at +4°C